SCHEMBL435757

SCHEMBL435757

Clc1ccc(-c2[c]cccc2Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
AHR P35869 2/20 0.37
LMNA P02545 3/20 0.35
CYP2A6 P11509 1/20 0.35
ALOX5 P09917 1/20 0.34
TSHR P16473 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
NFKB1 P19838 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SENP8 Q96LD8 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
NOTUM Q6P988 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790399 0.84 CYP2A6 (0.44) CYP1A2LMNACYP2A6TSHRKDM4E
SCHEMBL2012242 0.83 MAPK1 (0.38) LMNATSHRNPC1TP53RAB9A
SCHEMBL5899212 0.83 HPGD (0.35) KDM4EALDH1A1NPC1RAB9AHSD17B10
SCHEMBL10765346 0.83 NPC1 (0.44) CYP1A2AHRCYP2A6TSHRKDM4E
SCHEMBL4653269 0.81 CYP1A2 (0.39) CYP1A2AHRLMNACYP2A6ALOX5
SCHEMBL435279 0.79 CYP1A2 (0.38) CYP1A2AHRLMNACYP2A6ALOX5
SCHEMBL7733237 0.79 CYP1A2 (0.38) CYP1A2LMNACYP2A6ALOX5TSHR
SCHEMBL9265689 0.79 CYP1A2 (0.38) CYP1A2AHRLMNACYP2A6ALOX5
SCHEMBL8371280 0.79 CYP1A2 (0.38) CYP1A2AHRLMNACYP2A6ALOX5
SCHEMBL16720201 0.79 ALOX5 (0.45) CYP1A2LMNACYP2A6ALOX5TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8026085-B2 Methods and systems for selective fluorination of organic molecules CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2011-09-27 US claimed
EP-0414299-B1 Biocidal azoxime compounds SHELL INT RESEARCH (NL) 1994-06-15 EP claimed
EP-2912178-B1 SUPER-ENHANCERS AND METHODS OF USE THEREOF WHITEHEAD INST BIOMEDICAL RES (US) 2020-06-17 EP disclosed
EP-2912178-A1 SUPER-ENHANCERS AND METHODS OF USE THEREOF The Whitehead Institute for Biomedical Research (US) 2015-09-02 EP disclosed
WO-2014066848-A9 SUPER-ENHANCERS AND METHODS OF USE THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2014-08-14 WO disclosed
WO-2014066848-A1 SUPER-ENHANCERS AND METHODS OF USE THEREOF WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2014-05-01 WO disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
US-5459147-A Angeotensin-antagonistic effects; hypotensive, antiischemic, and antidiabetic agents, treating glaucoma DR. KARL THOMAE GMBH (DE) 1995-10-17 US disclosed
EP-0414299-B1 Biocidal azoxime compounds SHELL INT RESEARCH (NL) 1994-06-15 EP disclosed
EP-0363223-A2 3-Aryloxymethyl-cephalosporin derivatives, their preparation and their medical use Sankyo Company Limited (JP) 1990-04-11 EP disclosed
EP-0036834-B1 PROCESS FOR THE PREPARATION OF METAL COMPLEXES OF ISOINDOLINE AZINES CIBA-GEIGY AG (CH) 1983-12-07 EP disclosed
US-4405792-A Substituted pyridines and their preparation ETHYL CORPORATION (US) 1983-09-20 US disclosed
EP-0036834-A1 Process for the preparation of metal complexes of isoindoline azines CIBA-GEIGY AG (CH) 1981-09-30 EP disclosed
EP-0036387-A2 Process for the preparation of hydrazono-isoindolines CIBA-GEIGY AG (CH) 1981-09-23 EP disclosed
EP-0036388-A2 Isoindoline derivatives, process for their preparation and their use CIBA-GEIGY AG (CH) 1981-09-23 EP disclosed
US-3992416-A 4-Oxa-5-hydroxypolycycloalkenones-(3) BASF AKTIENGESELLSCHAFT (DT) 1976-11-16 US disclosed