SCHEMBL4359368

SCHEMBL4359368

CCCc1nn(Cc2ccccc2C(F)(F)F)c(=O)c(C(=O)NCC(=O)O)c1O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGLN3 Q9H6Z9 11/20 0.43
EGLN1 Q9GZT9 11/20 0.42
P2RY14 Q15391 1/20 0.41
AKR1B1 P15121 1/20 0.40
EGLN2 Q96KS0 7/20 0.40
CYSLTR2 Q9NS75 1/20 0.40
HIF1A Q16665 2/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359258 0.87 EGLN3 (0.47) EGLN3EGLN1EGLN2CYSLTR2
SCHEMBL4367648 0.86 EGLN1 (0.44) EGLN3EGLN1EGLN2HIF1A
SCHEMBL3852949 0.85 EGLN3 (0.48) EGLN3EGLN1P2RY14EGLN2CYSLTR2
SCHEMBL3847521 0.84 EGLN3 (0.43) EGLN3EGLN1P2RY14EGLN2CYSLTR2
SCHEMBL4358358 0.83 EGLN3 (0.45) EGLN3EGLN1AKR1B1EGLN2CYSLTR2
SCHEMBL4363076 0.83 EGLN1 (0.41) EGLN3EGLN1EGLN2HIF1A
SCHEMBL4356985 0.82 EGLN3 (0.43) EGLN3EGLN1EGLN2HIF1A
SCHEMBL4364331 0.81 HIF1A (0.43) EGLN3EGLN1AKR1B1HIF1A
SCHEMBL12727514 0.81 EGLN3 (0.59) EGLN3EGLN1EGLN2CYSLTR2HIF1A
SCHEMBL4359892 0.81 EGLN3 (0.59) EGLN3EGLN1EGLN2CYSLTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124565-A2 N-SUBSTITUTED GLYCINE DERIVATIVES: HYDROXYLASE INHIBITORS Smithkline Beecham Corporation (US) 2009-12-02 EP claimed
WO-2008089052-A2 N-SUBSTITUTED GLYCINE DERIVATIVES: HYDROXYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2008-07-24 WO claimed