SCHEMBL4360124

SCHEMBL4360124

CC1CN(C2(CNC(=O)c3cn(-c4ncccn4)c4cccc(Cl)c34)CCCCC2)CCN1C

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 12/20 0.51
HCN4 Q9Y3Q4 2/20 0.49
IL1B P01584 10/20 0.47
SLC6A9 P48067 4/20 0.42
HCN1 O60741 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13706816 1.00 P2RX7 (0.51) P2RX7HCN4IL1BSLC6A9HCN1
SCHEMBL4359934 0.91 HCN1 (0.42) P2RX7HCN4SLC6A9HCN1
SCHEMBL13706728 0.91 HCN1 (0.42) P2RX7HCN4SLC6A9HCN1
SCHEMBL3688404 0.89 HCN4 (0.63) P2RX7HCN4IL1BSLC6A9HCN1
SCHEMBL4357339 0.89 HCN4 (0.63) P2RX7HCN4IL1BSLC6A9HCN1
SCHEMBL13706815 0.88 P2RX7 (0.48) P2RX7HCN4IL1BHCN1
SCHEMBL13706899 0.88 P2RX7 (0.48) P2RX7HCN4IL1BHCN1
SCHEMBL4364179 0.88 P2RX7 (0.48) P2RX7HCN4IL1BHCN1
SCHEMBL13706897 0.88 P2RX7 (0.49) P2RX7HCN4IL1B
SCHEMBL4354322 0.87 P2RX7 (0.49) P2RX7HCN4IL1BSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO claimed