SCHEMBL4363213

SCHEMBL4363213

CNCC1=C(C(=O)O)c2ccccc2Oc2ccc(Cl)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
MEN1 O00255 2/20 0.41
PMP22 Q01453 2/20 0.41
KMT2A Q03164 2/20 0.41
ABCB11 O95342 1/20 0.41
LMNA P02545 1/20 0.41
CYP2C9 P11712 1/20 0.41
BLM P54132 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HRH4 Q9H3N8 4/20 0.39
HDAC3 O15379 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
HDAC4 P56524 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8170350 0.81 MAPK1 (0.48) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL10733451 0.73 MAPK1 (0.44) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL10729951 0.69 MAPK1 (0.50) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL10731007 0.69 MAPK1 (0.47) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL10730117 0.68 MAPK1 (0.49) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL19537683 0.67 MAPK1 (0.57) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL11266316 0.66 MAPK1 (0.53) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL2827619 0.66 LMNA (0.59) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL2829838 0.66 LMNA (0.59) MAPK1CYP1A2CYP3A4CYP2D6MEN1
SCHEMBL4847727 0.66 ALDH1A1 (0.41) MAPK1CYP1A2CYP3A4CYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1710241-B1 Intermediate compounds for the preparation of trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole ORGANON NV (NL) 2009-11-04 EP claimed