SCHEMBL4366546

SCHEMBL4366546

COc1ccc([C@H](CC(=O)O)N2CCC(CCCC3=CC=C4CCCNC4N3)C2=O)cn1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 19/20 0.45
ITGB3 P05106 18/20 0.45
ITGB6 P18564 5/20 0.45
ITGB1 P05556 3/20 0.45
ITGA2B P08514 3/20 0.45
ITGA5 P08648 2/20 0.45
ITGB8 P26012 2/20 0.45
ITGB5 P18084 1/20 0.37
ITGA4 P13612 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4366872 0.94 ITGAV (0.45) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL4368878 0.89 ITGAV (0.47) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL4047994 0.89 ITGAV (0.45) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL7592186 0.85 ITGAV (0.62) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL7594213 0.85 ITGAV (0.62) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL7557493 0.85 ITGAV (0.62) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL4386638 0.85 ITGB3 (0.43) ITGAVITGB3ITGB6ITGB1ITGA2B
SCHEMBL4370537 0.84 ITGB3 (0.65) ITGAVITGB3ITGA2BITGB5
SCHEMBL4363508 0.84 ITGB3 (0.65) ITGAVITGB3ITGA2BITGB5
SCHEMBL4372884 0.84 ITGB3 (0.65) ITGAVITGB3ITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP disclosed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP disclosed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed