SCHEMBL4366872

SCHEMBL4366872

CCOc1ccc([C@H](CC(=O)O)N2CCC(CCCC3=CC=C4CCCNC4N3)C2=O)cn1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 19/20 0.45
ITGB3 P05106 17/20 0.45
ITGB6 P18564 4/20 0.39
ITGB8 P26012 3/20 0.39
ITGB1 P05556 2/20 0.39
ITGA5 P08648 2/20 0.39
ITGA2B P08514 2/20 0.39
ITGB5 P18084 1/20 0.32
CHRNA7 P36544 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4366546 0.94 ITGAV (0.45) ITGAVITGB3ITGB6ITGB8ITGB1
SCHEMBL4368878 0.89 ITGAV (0.47) ITGAVITGB3ITGB6ITGB8ITGB1
SCHEMBL4047994 0.88 ITGAV (0.45) ITGAVITGB3ITGB6ITGB8ITGB1
SCHEMBL4376692 0.86 ITGB3 (0.44) ITGAVITGB3
SCHEMBL7589889 0.85 ITGAV (0.54) ITGAVITGB3ITGB6ITGB8ITGB1
SCHEMBL7554383 0.85 ITGAV (0.54) ITGAVITGB3ITGB6ITGB8ITGB1
SCHEMBL7594711 0.85 ITGAV (0.54) ITGAVITGB3ITGB6ITGB8ITGB1
SCHEMBL4386638 0.84 ITGB3 (0.43) ITGAVITGB3ITGB6ITGB8ITGB1
SCHEMBL4370537 0.83 ITGB3 (0.65) ITGAVITGB3ITGA2BITGB5
SCHEMBL4363508 0.83 ITGB3 (0.65) ITGAVITGB3ITGA2BITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1047425-A4 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2009-04-22 EP disclosed
EP-1047425-A1 INTEGRIN RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-11-02 EP disclosed
WO-1999030709-A1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1999-06-24 WO disclosed