SCHEMBL43672

SCHEMBL43672

N[C@H](C(=O)O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.52
CYP2D6 P10635 2/20 0.52
SRC P12931 1/20 0.52
LMNA P02545 2/20 0.50
MAPK1 P28482 1/20 0.50
SLC1A2 P43004 4/20 0.48
SLC1A3 P43003 3/20 0.48
SLC1A1 P43005 3/20 0.48
F2 P00734 1/20 0.46
GRM2 Q14416 1/20 0.46
GRM3 Q14832 1/20 0.46
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
ALOX5 P09917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL502830 1.00 DPP4 (0.52) DPP4CYP2D6SRCLMNAMAPK1
SCHEMBL43670 1.00 DPP4 (0.52) DPP4CYP2D6SRCLMNAMAPK1
SCHEMBL29360215 0.98 DPP4 (0.50) DPP4CYP2D6SRCLMNAMAPK1
Hydrochloric Acid SCHEMBL4799572 0.98 DPP4 (0.50) DPP4CYP2D6SRCLMNAMAPK1
Hydrochloric Acid SCHEMBL7582981 0.98 DPP4 (0.50) DPP4CYP2D6SRCLMNAMAPK1
Hydrochloric Acid SCHEMBL9445669 0.98 DPP4 (0.50) DPP4CYP2D6SRCLMNAMAPK1
Methane SCHEMBL29238636 0.98 DPP4 (0.50) DPP4CYP2D6SRCLMNAMAPK1
Carbamic Acid SCHEMBL29625257 0.96 CYP2D6 (0.48) DPP4CYP2D6SRCLMNAMAPK1
SCHEMBL7103757 0.88 LMNA (0.45) DPP4CYP2D6SRCLMNAMAPK1
Trifluoroacetic Acid SCHEMBL918979 0.88 SLC1A3 (0.44) DPP4CYP2D6SRCLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2881 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4719498-A1 RADIOLIGANDS FOR TARGETING CELL SURFACE RECEPTORS AND USES THEREOF Full-Life Technologies UK Limited (GB) 2026-04-08 EP claimed
EP-4719486-A1 CONJUGATES AND USES THEREOF Full-Life Technologies UK Limited (GB) 2026-04-08 EP claimed
US-12540161-B2 Linkers BICYCLETX LIMITED (GB) 2026-02-03 US claimed
US-20250339569-A1 CARBONIC ANHYDRASE IX LIGANDS 3B PHARMACEUTICALS GMBH (DE) 2025-11-06 US claimed
US-20250332223-A1 GHRH ANTAGONISTS FOR USE IN A METHOD OF TREATING SARCOIDOSIS UNIV MIAMI (US) 2025-10-30 US claimed
US-20250277012-A1 CONJUGATED HEPCIDIN MIMETICS PROTAGONIST THERAPEUTICS, INC. 2025-09-04 US claimed
US-20250250298-A1 ONCOLYTIC PEPTIDE AND USE THEREOF RISE BIOPHARMACEUTICALS INC. (CN) 2025-08-07 US claimed
US-12377135-B2 GHRH antagonists for use in a method of treating sarcoidosis UNIVERSITY OF MIAMI (US) 2025-08-05 US claimed
US-20250186539-A2 METHODS FOR TREATING CANCER BICYCLETX LIMITED (GB) 2025-06-12 US claimed
US-20250171776-A1 NON-CANONICAL CELL-PENETRATING PEPTIDES FOR ANTISENSE OLIGOMER DELIVERY SAREPTA THERAPEUTICS, INC. (US) 2025-05-29 US claimed
WO-2004056871-A2 PEPTIDES AND THEIR USE FOR THE TREATMENT OF HIV INFECTIONS IPF PHARMACEUTICALS GMBH (DE) 2004-07-08 WO claimed
US-6653295-B2 Protease inhibitor; viricide BRISTOL-MYERS SQUIBB COMPANY 2003-11-25 US claimed
WO-2003064458-A2 NOVEL PEPTIDE DERIVATIVES, PREPARATION AND THERAPEUTIC AND COSMETIC APPLICATION THEREOF INSTITUT EUROPEEN DE BIOLOGIE CELLULAIRE (FR) 2003-08-07 WO claimed
US-20030100768-A1 Imidazolidinones and their related derivatives as hepatitis C virus NS3 protease inhibitors BRISTOL-MYERS SQUIBB COMPANY (FORMERLY D/B/A DUPONT PHARMACEUTICALS COMPANY) 2003-05-29 US claimed
US-20030064962-A1 Inhibitors of hepatitis C virus NS3 protease BRISTOL-MYERS SQUIBB COMPANY (FORMERLY D/B/A DUPONT PHARMACEUTICALS COMPANY) 2003-04-03 US claimed
US-20020177725-A1 Peptide inhibitors of hepatitis C virus NS3 protein BRISTOL-MYERS SQUIBB COMPANY (FORMERLY D/B/A DUPONT PHARMACEUTICALS COMPANY) 2002-11-28 US claimed
WO-2002048116-A2 INHIBITORS OF HEPATITIS C VIRUS NS3 PROTEASE BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-06-20 WO claimed
WO-2002048157-A2 IMIDAZOLIDINONES AND THEIR RELATED DERIVATIVES AS HEPATITIS C VIRUS NS3 PROTEASE INHIBITORS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-06-20 WO claimed
WO-1993015042-A1 PROCESS FOR THE PREPARATION OF D(-) AND L(+)-3,3-DIPHENYLALANINE AND D(-) AND L(+)-SUBSTITUTED 3,3-DIPHENYLALANINES AND DERIVATIVES THEREOF WARNER-LAMBERT COMPANY (US) 1993-08-05 WO claimed
US-5198548-A Chemical intermediates for angiotensins WARNER-LAMBERT COMPANY (US) 1993-03-30 US claimed