SCHEMBL436731

SCHEMBL436731

Cc1cc(C)c2nc(C)cc(N)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.56
ALDH1A1 P00352 5/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
POLB P06746 3/20 0.56
RAD52 P43351 3/20 0.56
KMT2A Q03164 3/20 0.56
LMNA P02545 2/20 0.56
HTT P42858 2/20 0.56
HPGD P15428 2/20 0.56
MITF O75030 1/20 0.56
RAB9A P51151 1/20 0.47
NR4A2 P43354 2/20 0.47
TDP1 Q9NUW8 2/20 0.46
PARP1 P09874 1/20 0.44
NCF1 P14598 1/20 0.44
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GAA P10253 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11810566 0.81 KDM4E (0.56) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL436019 0.81 NR4A2 (0.53) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL442077 0.81 NR4A2 (0.45) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL442131 0.81 NR4A2 (0.45) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL440270 0.81 NR4A2 (0.62) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL11640984 0.76 KDM4E (0.59) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL17502194 0.76 LMNA (0.52) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL438224 0.74 NR4A2 (0.69) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL6088099 0.73 SMN1; SMN2 (0.43) KDM4EALDH1A1SMN1; SMN2POLBRAD52
SCHEMBL3120572 0.72 KDM4E (1.00) KDM4EALDH1A1SMN1; SMN2POLBRAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed
WO-2016022626-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed
US-20120065166-A1 Bone Modulators And Methods Therewith ESPINA VIRGINIA (US) 2012-03-15 US disclosed