Tebufelone

Tebufelone

SCHEMBL43674

C#CCCCC(=O)c1cc(C(C)(C)C)c(O)c(C(C)(C)C)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 1.00
PTGS1 P23219 6/20 1.00
ALOX5 P09917 5/20 1.00
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
LMNA P02545 2/20 0.45
RECQL P46063 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HTT P42858 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
MAPK1 P28482 1/20 0.42
F2R P25116 2/20 0.40
GAA P10253 2/20 0.39
GALR3 O60755 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7696046 0.95 PTGS2 (0.91) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL9420125 0.94 PTGS2 (0.89) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL7704620 0.94 PTGS2 (0.89) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL9860963 0.92 PTGS2 (0.85) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL9860870 0.92 PTGS2 (0.84) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL7701417 0.91 ALOX5 (0.83) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL10551397 0.87 PTGS2 (0.76) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL10551484 0.85 PTGS2 (0.73) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL9860910 0.85 PTGS2 (0.73) PTGS2PTGS1ALOX5KMT2AMEN1
SCHEMBL10548270 0.83 PTGS2 (0.70) PTGS2PTGS1ALOX5KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3846 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
WO-2023212179-A2 THERAPEUTIC COMPOSITIONS FOR SKIN DISORDERS AND WOUND REPAIR UNIVERSITY OF MIAMI (US) 2023-11-02 WO claimed
EP-3998932-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS Parsons, C. Lowell (US) 2022-05-25 EP claimed
US-20220110979-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC 2022-04-14 US claimed
EP-3908297-A1 FIBROBLAST REGENERATIVE CELLS Figene, LLC (US) 2021-11-17 EP claimed
EP-3279663-B1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES BRIGHAM & WOMENS HOSPITAL INC (US) 2021-07-28 EP claimed
WO-2021011566-A1 ALKALIZATION OF URINARY BLADDER WALL PRIOR TO TREATMENT WITH INTRAVESICAL HEPARIN AND ALKALINIZED LIDOCAINE TO ENHANCE RELIEF OF BLADDER PAIN SYMPTOMS PARSONS C LOWELL (US) 2021-01-21 WO claimed
CN-107085113-B Use of gelsolin for diagnosis and treatment of inflammatory diseases 布赖汉姆妇女医院有限公司 2020-07-17 CN claimed
WO-2020146874-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC (US) 2020-07-16 WO claimed
EP-3609483-A1 ARTICLE OF MANUFACTURE COMPRISING LOCAL ANESTHETIC, BUFFER, AND GLYCOSAMINOGLYCAN IN SYRINGE WITH IMPROVED STABILITY Urigen Pharmaceuticals, Inc. (US) 2020-02-19 EP claimed
WO-1994000130-A1 COMPOSITIONS FOR THE TREATMENT OF ARTHRITIS CONTAINING PHOSPHONATES AND NSAIDS PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1994-01-06 WO claimed
WO-1993023022-A1 SOLID DISPERSION COMPOSITIONS OF TEBUFELONE THE PROCTER & GAMBLE COMPANY (US) 1993-11-25 WO claimed
US-5189066-A Antiinflammatory agent THE PROCTER & GAMBLE COMPANY (US) 1993-02-23 US claimed
EP-0431659-A1 Pharmaceutical compositions of tebufelone THE PROCTER & GAMBLE COMPANY (US) 1991-06-12 EP claimed
EP-0251408-B1 NOVEL ANTI-INFLAMMATORY AGENTS, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR REDUCING INFLAMMATION THE PROCTER & GAMBLE COMPANY (US) 1991-04-17 EP claimed
US-4954332-A TOPICAL SUNSCREEN AGENTS; ULTRAVIOLET RADIATION AND OXIDATION RESISTNCE THE PROCTER & GAMBLE COMPANY (US) 1990-09-04 US claimed
US-4946671-A SUNSCREEN AGENTS THE PROCTER & GAMBLE COMPANY (US) 1990-08-07 US claimed
US-4847069-A SUNSCREEN AGENTS THE PROCTER & GAMBLE COMPANY (US) 1989-07-11 US claimed
US-4847071-A SUNSCREEN AGENTS THE PROCTER & GAMBLE COMPANY (US) 1989-07-11 US claimed
US-4708966-A SUBSTITUTED DI-TERT-BUTYL PHENOL DERIVATIVES THE PROCTER & GAMBLE COMPANY (US) 1987-11-24 US claimed