SCHEMBL4368719

SCHEMBL4368719

Cc1ccc(C(C)N)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
TDP1 Q9NUW8 4/20 0.50
CASP1 P29466 1/20 0.50
CYP3A4 P08684 5/20 0.46
ADRB2 P07550 1/20 0.43
GAA P10253 2/20 0.42
MAPT P10636 2/20 0.42
ALOX12 P18054 1/20 0.42
HTT P42858 1/20 0.42
HIF1A Q16665 1/20 0.42
LMNA P02545 1/20 0.40
TSHR P16473 3/20 0.39
TRPA1 O75762 1/20 0.39
PTGS1 P23219 1/20 0.39
CACNA1C Q13936 1/20 0.39
MAPK1 P28482 1/20 0.39
USP2 O75604 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16392261 1.00 ALDH1A1 (0.50) ALDH1A1TDP1CASP1CYP3A4ADRB2
Hydrochloric Acid SCHEMBL16370334 0.98 ALDH1A1 (0.48) ALDH1A1TDP1CASP1CYP3A4ADRB2
Hydrochloric Acid SCHEMBL16370328 0.98 ALDH1A1 (0.48) ALDH1A1TDP1CASP1CYP3A4ADRB2
Hydrochloric Acid SCHEMBL16370133 0.98 ALDH1A1 (0.48) ALDH1A1TDP1CASP1CYP3A4ADRB2
SCHEMBL512377 0.84 ALDH1A1 (0.59) ALDH1A1TDP1CASP1CYP3A4GAA
SCHEMBL11804318 0.82 ALDH1A1 (0.50) ALDH1A1TDP1CASP1CYP3A4GAA
Hydrochloric Acid SCHEMBL11333307 0.82 ALDH1A1 (0.57) ALDH1A1TDP1CASP1CYP3A4GAA
SCHEMBL13128971 0.81 ADRB2 (0.46) ALDH1A1TDP1ADRB2MAPTHIF1A
SCHEMBL13877347 0.81 ADRB2 (0.46) ALDH1A1TDP1ADRB2MAPTHIF1A
SCHEMBL3650358 0.81 ADRB2 (0.46) ALDH1A1TDP1ADRB2MAPTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015004481-A1 IMIDAZO-CONDENSED BICYCLES AS INHIBITORS OF DISCOIDIN DOMAIN RECEPTORS (DDRS) ASTEX THERAPEUTICS LIMITED (GB) 2015-01-15 WO disclosed
WO-2015004481-A1 IMIDAZO-CONDENSED BICYCLES AS INHIBITORS OF DISCOIDIN DOMAIN RECEPTORS (DDRS) ASTEX THERAPEUTICS LIMITED (GB) 2015-01-15 WO disclosed
WO-2009012375-A2 SQUARATE KINASE INHIBITORS WYETH (US) 2009-01-22 WO disclosed