SCHEMBL4373886

SCHEMBL4373886

COc1cccc(-c2cncnc2Oc2ccc3nc(NC(=O)Cc4ccccc4)sc3c2)c1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 7/20 0.64
WNT3A P56704 9/20 0.61
CYP3A4 P08684 1/20 0.58
MET P08581 1/20 0.56
ROCK2 O75116 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13587172 0.87 WNT3A (0.67) CSNK1DWNT3ACYP3A4MET
SCHEMBL4374930 0.83 MET (0.57) CSNK1DWNT3ACYP3A4METROCK2
SCHEMBL4914800 0.82 CSNK1D (0.87) CSNK1DWNT3ACYP3A4
SCHEMBL17287824 0.79 CSNK1D (1.00) CSNK1DWNT3ACYP3A4
SCHEMBL4371744 0.78 MET (0.77) CSNK1DWNT3AMETROCK2
SCHEMBL1723591 0.76 WNT3A (1.00) CSNK1DWNT3ACYP3A4
SCHEMBL17287785 0.76 CSNK1D (1.00) CSNK1DWNT3ACYP3A4
SCHEMBL17287645 0.76 CSNK1D (1.00) CSNK1DWNT3A
SCHEMBL4382502 0.75 MET (0.56) CSNK1DWNT3AMETROCK2
SCHEMBL4381371 0.74 MET (0.55) CSNK1DWNT3ACYP3A4METROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7626030-B2 Compounds and methods of use AMGEN INC. (US) 2009-12-01 US disclosed
US-20050245547-A1 6-((6,7-Bis(methoxy)-4-quinolinyl)oxy)-N-(3-methylphenyl)-1-benzofuran-3-carboxamide;antiproliferative; -metastasis; -carcinogenic; -tumor; -inflammatory; -arthritic agents;hypotensive agents; myocardium necrosis; rheumatic diseases; tyrosine kinase inhibitors; antiallergens; asthma AMGEN INC. 2005-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245547-A1 6-((6,7-Bis(methoxy)-4-quinolinyl)oxy)-N-(3-methylphenyl)-1-benzofuran-3-carboxamide;antiproliferative; -metastasis; -carcinogenic; -tumor; -inflammatory; -arthritic agents;hypotensive agents; myocardium necrosis; rheumatic diseases; tyrosine kinase inhibitors; antiallergens; asthma HGF, MET, HGFAC CSNK1D 1568/4885WNT3A 1795/4885CYP3A4 1110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.