SCHEMBL4373972

SCHEMBL4373972

CNc1ccc(Br)cc1C(=O)Nc1cc2c(cc1O)N(C(C)=O)C(C)(C)C(c1ccccc1)C2C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
TSHR P16473 1/20 0.35
AKR1C4 P17516 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
AKR1C1 Q04828 1/20 0.34
HCRTR1 O43613 3/20 0.34
HCRTR2 O43614 3/20 0.34
ALDH1A1 P00352 1/20 0.33
SORT1 Q99523 2/20 0.32
TP53 P04637 1/20 0.32
LMNA P02545 1/20 0.32
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
KMT2A Q03164 1/20 0.32
MAPK1 P28482 1/20 0.32
PTGFR P43088 1/20 0.31
DNMT3A Q9Y6K1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3527025 0.74 FSHR (0.56) TSHRNPSR1KMT2A
SCHEMBL4373967 0.73 TSHR (0.34) MAPTTSHRAKR1C4AKR1C3AKR1C2
SCHEMBL3525924 0.73 GAA (0.34) MAPTTSHRHCRTR1HCRTR2ALDH1A1
SCHEMBL1322915 0.64 FSHR (0.69) TSHRNPSR1KMT2A
SCHEMBL3524786 0.64 MAPT (0.42) MAPTALDH1A1TP53LMNAPOLB
SCHEMBL1323012 0.61 APEX1 (0.58) MAPTAKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL4367941 0.59 FSHR (0.64) TSHRNPSR1KMT2A
SCHEMBL28530907 0.59 ALDH1A1 (0.51) MAPTAKR1C3AKR1C2ALDH1A1LMNA
SCHEMBL224447 0.58 HCRTR1 (0.36) MAPTTSHRHCRTR1HCRTR2TP53
SCHEMBL336750 0.57 MAPT (0.68) MAPTAKR1C4AKR1C3AKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578726-B1 TETRAHYDROQUINOLINE DERIVATIVES ORGANON NV (NL) 2009-02-25 EP disclosed