SCHEMBL4374306

SCHEMBL4374306

CCOc1ccccc1-c1ccc2c(n1)N=C(N)N(C)C2N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.41
ALDH1A1 P00352 4/20 0.37
PDE3A Q14432 1/20 0.37
ENPP1 P22413 2/20 0.36
KDM4E B2RXH2 2/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
ENPP3 O14638 1/20 0.36
PTPRC P08575 1/20 0.36
NR3C1 P04150 1/20 0.35
TLR4 O00206 1/20 0.35
TLR3 O15455 1/20 0.35
TLR5 O60602 1/20 0.35
TLR2 O60603 1/20 0.35
CAMK2B Q13554 1/20 0.35
CAMK2G Q13555 1/20 0.35
CAMK2D Q13557 1/20 0.35
CAMK1 Q14012 1/20 0.35
CAMK4 Q16566 1/20 0.35
PNCK Q6P2M8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3745485 0.88 BRD4 (0.46) TLR4TLR3TLR5TLR2CAMK2B
SCHEMBL3729445 0.87 HSP90AA1 (0.41) DHFRALDH1A1KDM4ETLR8ADORA2A
SCHEMBL4377822 0.84 MAP4K1 (0.38) DHFRALDH1A1SCN9A
SCHEMBL4376393 0.84 HSP90AA1 (0.35) DHFRALDH1A1
SCHEMBL4384579 0.81 PTPN1 (0.37) TLR8GRM5SCN9A
SCHEMBL3734163 0.81 PTPN1 (0.37) KDM4ETSHRTLR8ADORA2AHSD17B10
SCHEMBL3739137 0.80 HSD17B10 (0.38) ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3727477 0.80 PTPN1 (0.38) ALDH1A1TLR8ADORA2AADORA1
SCHEMBL3734730 0.77 PTPN1 (0.41) TLR8SCN9A
SCHEMBL3737667 0.76 ASIC3 (0.40) ALDH1A1KDM4EPKMTLR8ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910359-B1 PYRIDO [2 , 3-D]PYRIMIDINE-2 , 4-DIAMINE COMPOUNDS AS PTPlB INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-18 EP claimed