SCHEMBL4377822

SCHEMBL4377822

CCOc1cccc(F)c1-c1ccc2c(n1)N=C(N)N(C)C2N

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 4/20 0.38
SCN9A Q15858 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
HCRTR1 O43613 6/20 0.33
HCRTR2 O43614 6/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KLKB1 P03952 1/20 0.32
RPS6KA2 Q15349 1/20 0.32
IKBKB O14920 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ATM Q13315 1/20 0.31
SSTR5 P35346 1/20 0.30
KCNH2 Q12809 1/20 0.30
DHFR P00374 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387064 0.88 MAP4K1 (0.40) MAP4K1RPS6KA2
SCHEMBL4376393 0.87 HSP90AA1 (0.35) L3MBTL1IKBKBALDH1A1DHFR
SCHEMBL4384579 0.87 PTPN1 (0.37) SCN9AIKBKB
SCHEMBL3727498 0.86 F2RL3 (0.33)
SCHEMBL4384578 0.85 ALOX5AP (0.35) MAP4K1RPS6KA2
SCHEMBL4374306 0.84 DHFR (0.41) SCN9AALDH1A1DHFR
SCHEMBL4386872 0.82 MCHR1 (0.36) MAP4K1
SCHEMBL3734371 0.81 PDE2A (0.32) MAP4K1
SCHEMBL3732360 0.79 PTPN1 (0.45) SCN9A
SCHEMBL4386942 0.77 PTPN1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910359-B1 PYRIDO [2 , 3-D]PYRIMIDINE-2 , 4-DIAMINE COMPOUNDS AS PTPlB INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-18 EP claimed