SCHEMBL4374699

SCHEMBL4374699

CN1CCN(c2cccc(C(F)(F)F)c2-c2ccc3c(n2)N=C(N)N(C)C3N)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 3/20 0.44
HRH4 Q9H3N8 2/20 0.37
ADRA2C P18825 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
CYP1A2 P05177 4/20 0.34
CYP2C19 P33261 3/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2D6 P10635 3/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAPK1 P28482 2/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
CCNA1 P78396 2/20 0.33
CDK4 P11802 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3732060 0.92 PTPN1 (0.52) PTPN1HTR2AHTR2CHTR2BGSK3B
SCHEMBL4381212 0.92 PTPN1 (0.43) PTPN1CYP1A2CYP2C19ALDH1A1TSHR
SCHEMBL4374330 0.91 PTPN1 (0.42) PTPN1HTR2AHTR2CHTR2BKDM4E
SCHEMBL4376462 0.91 PTPN1 (0.42) PTPN1HTR2AHTR2CHTR2BGSK3B
SCHEMBL4374731 0.90 PTPN1 (0.54) PTPN1HTR2BKDM4EALDH1A1GSK3B
SCHEMBL4389725 0.88 PTPN1 (0.43) PTPN1CYP1A2CYP2D6KDM4EALDH1A1
SCHEMBL4381688 0.88 HSD11B1 (0.43) PTPN1HTR2AHTR2CKDM4EALDH1A1
SCHEMBL4382742 0.87 HRH4 (0.42) PTPN1HRH4ADRA2CALDH1A1MAPK1
SCHEMBL3742273 0.86 PTPN1 (0.36) PTPN1HTR2AHTR2CHTR2B
SCHEMBL4378466 0.86 PTPN1 (0.39) PTPN1HTR2ACYP3A4TSHRDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910359-B1 PYRIDO [2 , 3-D]PYRIMIDINE-2 , 4-DIAMINE COMPOUNDS AS PTPlB INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-18 EP claimed