SCHEMBL4374944

SCHEMBL4374944

COc1ccc2c(c1)c(CCOS(=O)(=O)c1ccc(C)cc1)c(C)n2S(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 11/20 0.60
PTGDR2 Q9Y5Y4 3/20 0.52
PTGDR Q13258 1/20 0.52
MAPT P10636 1/20 0.43
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
PTGES O14684 1/20 0.41
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18239754 0.81 HTR6 (0.57) HTR6PTGDR2PTGDR
SCHEMBL18239786 0.79 HTR6 (0.56) HTR6PTGDR2PTGDRMAPTPTGS1
SCHEMBL18222517 0.79 HTR6 (0.56) HTR6PTGDR2PTGDR
SCHEMBL4374940 0.75 HTR6 (0.49) HTR6PTGDR2PTGDRMAPTPTGS1
SCHEMBL5498898 0.75 HTR6 (1.00) HTR6PTGDR2PTGDR
SCHEMBL3566087 0.74 HTR6 (0.60) HTR6PTGDR2PTGDR
SCHEMBL18317950 0.74 CA12 (0.43) MAPT
Oxalic Acid SCHEMBL7448579 0.74 HTR6 (0.71) HTR6PTGDR2PTGDR
SCHEMBL12628490 0.73 HTR6 (0.56) HTR6PTGDR2PTGDRMAPTPTGS1
SCHEMBL1429408 0.72 MEN1 (0.45) HTR6ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006089-A2 A2 ADENOSINE RECEPTOR AGONISTS GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2009-01-08 WO disclosed