SCHEMBL4375376

SCHEMBL4375376

CCOc1cc(C)nc(F)c1OC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.39
DHFR P00374 1/20 0.39
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HSD17B10 Q99714 2/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
PKM P14618 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPK1 P28482 1/20 0.37
LMNA P02545 1/20 0.36
MAPT P10636 2/20 0.36
SYK P43405 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13743050 0.82 AGTR1 (0.43) TUBB1DHFRNCOA1NCOA3MEN1
SCHEMBL4376433 0.71 HPGD (0.44) TUBB1MEN1KMT2AKDM4EHPGD
SCHEMBL2085154 0.71 KDM4E (0.43) MEN1KMT2AHSD17B10KDM4EHPGD
SCHEMBL14432911 0.71 PTGS2 (0.50) TUBB1DHFRNCOA1NCOA3MEN1
SCHEMBL4378885 0.68 KDM4E (0.30) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL20676684 0.67 KDM4E (0.46) DHFRKDM4EMAPK1MAPTTSHR
SCHEMBL21823706 0.67 NCOA1 (0.45) TUBB1NCOA1NCOA3MEN1KMT2A
SCHEMBL9804771 0.66 CYP3A4 (0.64) TUBB1DHFRNCOA1NCOA3HSD17B10
SCHEMBL1731146 0.66 NCOA1 (0.48) TUBB1NCOA1NCOA3MEN1KMT2A
SCHEMBL18310639 0.64 KMT2A (0.36) MEN1KMT2AHSD17B10KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103950-A1 FLUORINATED PYRIDIN-4-0NES BTG INTERNATIONAL LIMITED (GB) 2009-08-27 WO disclosed
WO-2009103950-A1 FLUORINATED PYRIDIN-4-0NES BTG INTERNATIONAL LIMITED (GB) 2009-08-27 WO disclosed