SCHEMBL4377535

SCHEMBL4377535

COc1cc(-c2cccc(NS(C)(=O)=O)c2)ccc1C(=O)NNC(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 4/20 0.47
TGFBR1 P36897 1/20 0.47
ACVR1 Q04771 1/20 0.47
KIF11 P52732 1/20 0.45
POLB P06746 1/20 0.45
ADRB3 P13945 3/20 0.44
ADRB1 P08588 2/20 0.44
HSD17B1 P14061 2/20 0.44
HSD17B2 P37059 2/20 0.44
BRD4 O60885 2/20 0.44
IKBKB O14920 1/20 0.43
CHUK O15111 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
RAF1 P04049 1/20 0.43
BRAF P15056 1/20 0.43
POLQ O75417 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3139471 0.87 FYN (0.52) FYNTGFBR1ACVR1KIF11POLB
SCHEMBL3138802 0.86 FYN (0.44) FYNTGFBR1ACVR1KIF11POLB
SCHEMBL3137569 0.86 FYN (0.52) FYNTGFBR1ACVR1KIF11POLB
SCHEMBL3143232 0.84 POLB (0.57) FYNTGFBR1ACVR1KIF11POLB
SCHEMBL5359155 0.72 ALDH1A1 (0.53) FYNPOLBCYP1A2CYP3A4CYP2D6
SCHEMBL1308772 0.72 FYN (0.57) FYNTGFBR1ACVR1POLB
SCHEMBL13485182 0.71 POLB (0.71) KIF11POLBHSD17B1HSD17B2BRD4
SCHEMBL21092440 0.71 KIF11 (0.69) KIF11HSD17B1HSD17B2BRD4IKBKB
SCHEMBL2040073 0.71 KIF11 (0.61) KIF11POLBHSD17B1HSD17B2BRD4
SCHEMBL3100085 0.70 TUBB4A (0.48) FYNTGFBR1ACVR1HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119719-A1 THIAZEPINE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2009-11-18 EP disclosed