SCHEMBL4378574

SCHEMBL4378574

O=C(C=CN1CCN(C2CCCC2)CC1)c1cccc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.53
KDM4E B2RXH2 3/20 0.50
ALDH1A1 P00352 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HIF1A Q16665 1/20 0.50
SIGMAR1 Q99720 4/20 0.45
HRH3 Q9Y5N1 2/20 0.44
KCNH2 Q12809 1/20 0.44
GPR52 Q9Y2T5 1/20 0.42
KDM2B Q8NHM5 1/20 0.42
ACACB O00763 1/20 0.41
ACACA Q13085 1/20 0.41
TP53BP1 Q12888 2/20 0.41
L3MBTL3 Q96JM7 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
LMNA P02545 2/20 0.41
MBTD1 Q05BQ5 1/20 0.41
POLB P06746 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4376221 0.99 GAA (0.52) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL4384264 0.99 GAA (0.52) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL2829562 0.90 GAA (0.53) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL2833287 0.89 GAA (0.52) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL4382981 0.78 GAA (0.53) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL4377273 0.77 GPR52 (0.44) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL4375430 0.75 HRH3 (0.48) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL4378514 0.75 GPR52 (0.45) KDM4EALDH1A1MEN1KMT2AHRH3
SCHEMBL4375865 0.74 ALDH1A1 (0.50) KDM4EALDH1A1MEN1KMT2AHIF1A
SCHEMBL4377900 0.73 HRH3 (0.52) MEN1KMT2AHRH3GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1421071-B1 SUBSTITUTED PIPERAZINE AND DIAZEPANE DERIVAIVES AS HISTAMINE H3 RECEPTOR MODULATORS HIGH POINT PHARMACEUTICALS LLC (US) 2009-11-18 EP claimed
EP-1421071-B1 SUBSTITUTED PIPERAZINE AND DIAZEPANE DERIVAIVES AS HISTAMINE H3 RECEPTOR MODULATORS HIGH POINT PHARMACEUTICALS LLC (US) 2009-11-18 EP disclosed