SCHEMBL4378971

SCHEMBL4378971

COC(=O)CCc1ccncc1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.54
CDK8 P49336 1/20 0.54
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 3/20 0.51
GLA P06280 1/20 0.51
GAA P10253 1/20 0.51
AOC1 P19801 2/20 0.47
AOC3 Q16853 2/20 0.47
HDAC1 Q13547 1/20 0.44
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
KDM6B O15054 1/20 0.41
KDM4A O75164 1/20 0.41
THRB P10828 1/20 0.41
KDM4D Q6B0I6 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CYP11B1 P15538 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3651691 0.85 CYP4F2 (0.50) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL18808055 0.84 ALDH1A1 (0.54) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL27582108 0.83 CCNC (0.55) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL27224524 0.83 CCNC (0.55) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL8216031 0.82 AOC1 (0.52) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL19799358 0.81 CCNC (0.54) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL15773725 0.81 CCNC (0.54) CCNCCDK8ALDH1A1KDM4EMAPT
SCHEMBL2999880 0.80 AOC1 (0.53) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL19838578 0.77 ALDH1A1 (0.54) CCNCCDK8ALDH1A1KDM4EGLA
SCHEMBL29792765 0.77 ALDH1A1 (0.54) CCNCCDK8ALDH1A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2083011-B1 PYRROLINE DERIVATIVES AGAINST CELL RELEASING TUMOR NECROSIS FACTOR, PREPARATION METHODS AND USES THEREOF TIANJIN HEMAY BIO TECH CO LTD (CN) 2014-06-04 EP disclosed
CN-101186612-B Pyrroline derivative capable of inhibiting cell to release tumor necrotic factor and its preparation and application TIANJIN HEMEI BIOLOG TECHNOLOGY CO LTD 2012-10-03 CN disclosed
EP-2083011-A1 PYRROLINE DERIVATIVES AGAINST CELL RELEASING TUMOR NECROSIS FACTOR, PREPARATION METHODS AND USES THEREOF Tian Jin Hemay Bio-Tech Co., Ltd. (CN) 2009-07-29 EP disclosed
CN-101186612-A Pyrroline derivative capable of inhibiting cell to release tumor necrotic factor and its preparation and application TIANJIN HEMEI BIOLOG TECHNOLOG (CN) 2008-05-28 CN disclosed
CN-1320125-A Trizolopyridines for the treamtent of thrombosis disorders ORTHO MCNEIL PHARM INC (US) 2001-10-31 CN disclosed