SCHEMBL4380045

SCHEMBL4380045

C=C(C(=O)OC)c1ccc2c(c1)CNCC2

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MELK Q14680 2/20 0.48
PNMT P11086 4/20 0.45
SLC2A1 P11166 1/20 0.44
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30745003 0.82 MELK (0.52) MELKPNMTSLC2A1ADRA2AADRA2B
SCHEMBL308122 0.82 MELK (0.52) MELKPNMTSLC2A1ADRA2AADRA2B
Hydrochloric Acid SCHEMBL29903254 0.81 MELK (0.51) MELKPNMTSLC2A1ADRA2AADRA2B
Hydrochloric Acid SCHEMBL1017102 0.81 MELK (0.51) MELKPNMTSLC2A1ADRA2AADRA2B
SCHEMBL4544279 0.81 MELK (0.48) MELKPNMTSLC2A1ADRA2AADRA2B
SCHEMBL3248558 0.77 MELK (0.56) MELKPNMTSLC2A1ADRA2AADRA2B
SCHEMBL29784680 0.77 ASIC3 (0.47) MELK
SCHEMBL1035136 0.77 ASIC3 (0.47) MELK
SCHEMBL1014888 0.77 MELK (0.56) MELKPNMTSLC2A1ADRA2AADRA2B
SCHEMBL4544259 0.76 ASIC3 (0.47) MELKPNMTSLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120910-A2 HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF Novartis Ag (CH) 2009-11-25 EP disclosed
WO-2008076954-A2 HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2008-06-26 WO disclosed