SCHEMBL4544279

SCHEMBL4544279

C=C(C(N)=O)c1ccc2c(c1)CNCC2

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MELK Q14680 1/20 0.48
PNMT P11086 6/20 0.48
ADRA2A P08913 3/20 0.48
ADRA2B P18089 2/20 0.48
ADRA2C P18825 2/20 0.48
SLC2A1 P11166 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4543801 0.94 PLAU (0.49) MELKPNMTADRA2AADRA2BADRA2C
Trifluoroacetic Acid SCHEMBL31335937 0.91 MELK (0.44) MELKPNMTADRA2AADRA2BADRA2C
SCHEMBL29728413 0.84 PNMT (0.53) MELKPNMTADRA2AADRA2BADRA2C
SCHEMBL1033504 0.84 PNMT (0.53) MELKPNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL17748278 0.83 PNMT (0.51) MELKPNMTADRA2AADRA2BADRA2C
SCHEMBL4380045 0.81 MELK (0.48) MELKPNMTADRA2AADRA2BADRA2C
SCHEMBL30357006 0.79 ALDH1A1 (0.59) ADRA2AADRA2BADRA2C
SCHEMBL29589725 0.79 ALDH1A1 (0.59) MELKPNMTADRA2AADRA2BADRA2C
SCHEMBL1026913 0.79 ALDH1A1 (0.59) MELKPNMTADRA2AADRA2BADRA2C
SCHEMBL1119301 0.78 PLAU (0.53) MELKPNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120910-A2 HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF Novartis Ag (CH) 2009-11-25 EP claimed
WO-2008076954-A2 HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF NOVARTIS AG (CH) 2008-06-26 WO claimed