SCHEMBL4380129

SCHEMBL4380129

COc1c(NC(c2ccccc2)(c2ccccc2)c2ccccc2)ccc2[nH]nc(-c3cccc(F)c3)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.43
MAP2K4 P45985 5/20 0.40
TTK P33981 1/20 0.39
FYN P06241 2/20 0.38
CLK2 P49760 3/20 0.37
CLK3 P49761 3/20 0.37
DYRK1A Q13627 3/20 0.37
LRRK2 Q5S007 3/20 0.35
MAPK8 P45983 1/20 0.35
MAPK10 P53779 1/20 0.35
MAPK14 Q16539 1/20 0.35
MAP2K7 O14733 1/20 0.35
TACR3 P29371 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859116 0.79 MAP2K4 (0.48) NTRK1MAP2K4TTKFYNLRRK2
SCHEMBL2863456 0.78 TTK (0.48) NTRK1MAP2K4TTKFYNCLK2
SCHEMBL2863072 0.77 TTK (0.47) NTRK1MAP2K4TTKFYNCLK2
SCHEMBL2864633 0.75 MAP2K4 (0.47) NTRK1MAP2K4TTKFYNLRRK2
SCHEMBL4327628 0.75 GSK3B (0.53) NTRK1CLK2DYRK1AGSK3AGSK3B
SCHEMBL2862698 0.74 NTRK1 (0.44) NTRK1MAP2K4TTKFYNCLK2
SCHEMBL2864166 0.74 NTRK1 (0.49) NTRK1MAP2K4TTKFYNCLK2
SCHEMBL4335949 0.71 CDK9 (0.44) NTRK1TTKCLK2CLK3DYRK1A
SCHEMBL13198269 0.71 MEN1 (0.41) NTRK1MAP2K4TTKDYRK1AGSK3A
SCHEMBL4335950 0.71 MEN1 (0.41) NTRK1MAP2K4TTKDYRK1AGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1380576-B1 1H-INDAZOLE COMPOUNDS INHIBITING JNK EISAI R&D MAN CO LTD (JP) 2009-11-25 EP disclosed