SCHEMBL4380885

SCHEMBL4380885

CCOc1ccc2c(c1)c(C(=O)C(=O)Nc1ccncn1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1.COc1ccc2c(c1)c(C(=O)C(=O)Nc1ccncn1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.45
PLA2G2A P14555 3/20 0.42
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
RGS12 O14924 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
PKM P14618 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
GNAI1 P63096 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
ALOX5 P09917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4088397 0.97 FAAH (0.43) FAAHPLA2G2AMAPTCYP3A4CYP2C9
SCHEMBL4088424 0.96 FAAH (0.47) FAAHPLA2G2AMAPTKMT2AMEN1
SCHEMBL4083416 0.88 F2RL3 (0.35) FAAHPLA2G2AMAPTKMT2AMEN1
SCHEMBL4094189 0.87 PLA2G2A (0.41) FAAHPLA2G2AMAPTKMT2AMEN1
SCHEMBL4088689 0.87 FAAH (0.44) FAAHKMT2ACYP3A4CYP2C9ALOX5
SCHEMBL2993129 0.87 FAAH (0.51) FAAHPLA2G2AMAPTLMNAALOX5
SCHEMBL2995166 0.87 FAAH (0.46) FAAHPLA2G2AMAPTKMT2AMEN1
SCHEMBL4095302 0.86 FAAH (0.48) FAAHPLA2G2AMAPTKMT2AMEN1
SCHEMBL4093742 0.86 FAAH (0.49) FAAHPLA2G2AMAPTKMT2AMEN1
SCHEMBL4562856 0.86 FAAH (0.53) FAAHMAPTKMT2AMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed