SCHEMBL4381736

SCHEMBL4381736

CC(=O)c1ccc2c(c1)CN(CCCSc1nnc(-c3ccccc3)n1C(C)C)CC2

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 18/20 0.47
DRD2 P14416 14/20 0.47
KCNH2 Q12809 11/20 0.47
HRH1 P35367 1/20 0.41
MAP3K5 Q99683 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PPARG P37231 1/20 0.40
KMT2A Q03164 1/20 0.40
NR2E3 Q9Y5X4 1/20 0.40
NCOR2 Q9Y618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387104 0.90 DRD3 (0.59) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4387400 0.87 DRD3 (0.48) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4380355 0.86 DRD3 (0.47) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4383491 0.86 DRD3 (0.47) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4385545 0.86 DRD3 (0.47) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4705240 0.82 DRD3 (0.58) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4701185 0.81 DRD3 (0.57) DRD3DRD2KCNH2HRH1KDM4E
SCHEMBL4703079 0.81 DRD3 (0.59) DRD3DRD2KCNH2ALDH1A1POLB
SCHEMBL4704001 0.79 DRD3 (0.55) DRD3DRD2KCNH2HRH1KDM4E
Oxalic Acid SCHEMBL7204441 0.79 DRD3 (0.55) DRD3DRD2KCNH2HRH1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP claimed