SCHEMBL4387400

SCHEMBL4387400

CCn1c(SCCCN2CCc3ccc(C(C)=O)cc3C2)nnc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 7/20 0.48
DRD2 P14416 6/20 0.48
KCNH2 Q12809 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 2/20 0.47
KDM4E B2RXH2 2/20 0.47
ALPL P05186 1/20 0.47
POLB P06746 1/20 0.47
ALPG P10696 1/20 0.47
ALOX12 P18054 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NPC1 O15118 1/20 0.46
PTK2 Q05397 1/20 0.44
HDAC2 Q92769 1/20 0.44
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
HRH1 P35367 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4380355 0.94 DRD3 (0.47) DRD3DRD2KCNH2SMN1; SMN2MAPT
SCHEMBL4385545 0.93 DRD3 (0.47) DRD3DRD2KCNH2SMN1; SMN2MAPT
SCHEMBL4387104 0.90 DRD3 (0.59) DRD3DRD2KCNH2MAPTKDM4E
SCHEMBL4381736 0.87 DRD3 (0.47) DRD3DRD2KCNH2MAPTKDM4E
SCHEMBL4383491 0.86 DRD3 (0.47) DRD3DRD2KCNH2MAPTKDM4E
SCHEMBL4701185 0.83 DRD3 (0.57) DRD3DRD2KCNH2MAPTGAA
SCHEMBL4705240 0.82 DRD3 (0.58) DRD3DRD2KCNH2MAPTKDM4E
SCHEMBL4703079 0.81 DRD3 (0.59) DRD3DRD2KCNH2POLBLMNA
SCHEMBL4704001 0.80 DRD3 (0.55) DRD3DRD2KCNH2MAPTKDM4E
SCHEMBL4386792 0.80 DRD3 (0.63) DRD3DRD2KCNH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144405-B1 TRIAZOLE COMPOUNDS WITH DOPAMINE-D3-RECEPTOR AFFINITY ABBOTT GMBH & CO KG (DE) 2009-11-25 EP claimed