SCHEMBL4383799

SCHEMBL4383799

CCC1(NC(=O)c2ccc(OC)nc2OC)CCCCn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 14/20 0.35
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
HPGD P15428 2/20 0.33
TSHR P16473 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HSD17B10 Q99714 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
CYP3A4 P08684 1/20 0.32
SIRT1 Q96EB6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387224 0.90 ALDH1A1 (0.36) GSK3BTSHRSMN1; SMN2ALDH1A1CYP3A4
SCHEMBL4387999 0.89 GSK3B (0.37) GSK3BRAB9ANPC1HPGDTSHR
SCHEMBL4384554 0.79 GSK3B (0.37) GSK3BTSHRALDH1A1CYP3A4
SCHEMBL4381292 0.77 GSK3B (0.41) GSK3BRAB9ANPC1CYP3A4
SCHEMBL4387202 0.76 GSK3B (0.41) GSK3BRAB9ANPC1CYP3A4
SCHEMBL4378591 0.76 GSK3B (0.38) GSK3BCYP3A4
SCHEMBL3373754 0.72 OPRD1 (0.41) GSK3BRAB9ANPC1CYP3A4
SCHEMBL2066100 0.72 GSK3B (0.43) GSK3BALDH1A1CYP3A4
SCHEMBL2065915 0.72 GSK3B (0.37) GSK3B
SCHEMBL3659041 0.72 GSK3B (0.45) GSK3BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP claimed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO claimed
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP disclosed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO disclosed