SCHEMBL4383908

SCHEMBL4383908

Clc1ccc(Cn2c[c]c3ccccc32)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.48
SIGMAR1 Q99720 1/20 0.46
DBH P09172 1/20 0.43
VDR P11473 1/20 0.43
KCNA3 P22001 1/20 0.43
LMNA P02545 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
ALOX12 P18054 1/20 0.42
CYP2D6 P10635 1/20 0.42
TSHR P16473 1/20 0.42
PMP22 Q01453 1/20 0.42
HIF1A Q16665 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29136178 0.88 DBH (0.46) SLC9A1SIGMAR1DBHKCNA3LMNA
SCHEMBL27889061 0.82 DBH (0.41) SLC9A1SIGMAR1DBHLMNACYP1A2
SCHEMBL27905750 0.80 HTT (0.49) SIGMAR1LMNACYP1A2CYP3A4CYP2C9
SCHEMBL15062690 0.79 IDO1 (0.39) DBHLMNAMAPTSMN1; SMN2
SCHEMBL694560 0.74 TNF (0.44) SLC9A1SIGMAR1DBHLMNAALDH1A1
SCHEMBL15062577 0.73 VDR (0.49) SLC9A1SIGMAR1VDRLMNACYP1A2
SCHEMBL29136175 0.73 SLC9A1 (0.58) SLC9A1SIGMAR1VDRLMNACYP1A2
SCHEMBL28261607 0.73 KCNA3 (0.53) SLC9A1SIGMAR1DBHVDRKCNA3
SCHEMBL15062502 0.71 LMNA (0.49) SLC9A1SIGMAR1VDRLMNACYP1A2
SCHEMBL20715687 0.71 CYP11B1 (0.66) SLC9A1VDRLMNATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117003739-A Nitrogen-containing heterocyclic compound, preparation method and application thereof 安徽中医药大学 2023-11-07 CN disclosed
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed