SCHEMBL4386508

SCHEMBL4386508

CCOc1ccc2c(c1)c(C(=O)C(=O)Nc1ncccn1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl.COc1ccc2c(c1)c(C(=O)C(=O)Nc1ncccn1)c(C(F)(F)F)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 6/20 0.40
EDNRB P24530 3/20 0.38
FAAH O00519 1/20 0.38
F2RL3 Q96RI0 1/20 0.37
PTGS2 P35354 2/20 0.37
ALOX5AP P20292 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4099175 0.97 ALOX5AP (0.38) PLA2G2AEDNRBFAAHF2RL3ALOX5AP
SCHEMBL4095857 0.96 PLA2G2A (0.42) PLA2G2AFAAHF2RL3PTGS2ALOX5AP
SCHEMBL3002874 0.90 PTGS2 (0.46) PLA2G2AEDNRBFAAHPTGS2LMNA
SCHEMBL3008455 0.89 MEN1 (0.42) PLA2G2AEDNRBFAAHLMNASMN1; SMN2
SCHEMBL3007424 0.89 NPC1 (0.38) PLA2G2AEDNRBFAAHF2RL3ALOX5AP
SCHEMBL4088892 0.88 EPHX2 (0.40) FAAHLMNASMN1; SMN2
SCHEMBL3001872 0.88 PLA2G2A (0.41) PLA2G2AFAAHF2RL3PTGS2PTGDR2
SCHEMBL4088383 0.88 FAAH (0.46) FAAHALOX5AP
SCHEMBL3005046 0.87 FAAH (0.41) FAAHF2RL3ALOX5APLMNASMN1; SMN2
SCHEMBL3008903 0.87 MEN1 (0.41) EDNRBF2RL3ALOX5APLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed