SCHEMBL4386586

SCHEMBL4386586

CCOC(=O)Oc1cc(OC(=O)OCC)c(-c2ccccc2)c(CCOCCOC)c1CC

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 9/20 0.37
TRPV1 Q8NER1 2/20 0.37
ALOX5 P09917 1/20 0.36
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TSHR P16473 1/20 0.35
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4389593 0.88 PDE4A (0.36) ADORA3ALOX5TP53SMN1; SMN2KDM4E
SCHEMBL4390309 0.85 NCEH1 (0.43) SMN1; SMN2NPC1ALDH1A1LMNARAB9A
SCHEMBL4385454 0.83 ALDH1A1 (0.34) ALOX5KDM4EALDH1A1MAPTHPGD
SCHEMBL4385095 0.81 ESR1 (0.36) ALDH1A1MAPT
SCHEMBL4395183 0.80 SMN1; SMN2 (0.38) TP53SMN1; SMN2KDM4ENPC1ALDH1A1
SCHEMBL4384143 0.79 KDM4E (0.36) KDM4EHPGD
SCHEMBL4382068 0.77 EGFR (0.35) TP53SMN1; SMN2MEN1KMT2A
SCHEMBL4384177 0.77 CNR2 (0.35) ALOX5ALDH1A1MAPTHPGDMEN1
SCHEMBL4386639 0.75 ESR1 (0.38) ALDH1A1MAPT
SCHEMBL4386523 0.74 RXRA (0.40) TP53KDM4EALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7538241-B2 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-05-26 US disclosed
US-20070155813-A1 Hsp90 family protein inhibitors KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-07-05 US disclosed
EP-1704856-A1 HSP90 FAMILY PROTEIN INHIBITOR KYOWA HAKKO KOGYO CO., LTD. (JP) 2006-09-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070155813-A1 Hsp90 family protein inhibitors HSP90AB1, HEATR1, HSP90AB2P ADORA3 3728/4885TRPV1 2108/4885ALOX5 4819/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.