SCHEMBL4386979

SCHEMBL4386979

O=C(NC1CCn2c1nc(-c1ccncn1)cc2=O)c1ccc2ncccc2n1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 14/20 0.38
CYP3A4 P08684 2/20 0.37
TNKS O95271 2/20 0.36
TNKS2 Q9H2K2 2/20 0.36
CYP2D6 P10635 2/20 0.36
NAMPT P43490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4384596 0.95 GSK3B (0.37) GSK3BCYP3A4TNKSTNKS2CYP2D6
SCHEMBL4383569 0.94 GSK3B (0.37) GSK3BCYP3A4TNKSTNKS2CYP2D6
SCHEMBL3403493 0.90 GSK3B (0.35) GSK3BCYP3A4TNKSTNKS2CYP2D6
SCHEMBL4387983 0.89 NAMPT (0.36) GSK3BNAMPT
SCHEMBL3664250 0.85 GSK3B (0.43) GSK3BCYP2D6
SCHEMBL4386475 0.83 HPGD (0.38) GSK3BNAMPT
SCHEMBL4385219 0.80 MEN1 (0.43) GSK3BCYP3A4CYP2D6
SCHEMBL4401406 0.78 GSK3B (0.37) GSK3BCYP3A4TNKSTNKS2CYP2D6
SCHEMBL4955066 0.78 GSK3B (0.37) GSK3BCYP3A4TNKSTNKS2CYP2D6
SCHEMBL4380168 0.77 GSK3B (0.38) GSK3BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP claimed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO claimed
EP-1939187-A1 Substituted heteroaryl pyridopyrimidone derivatives Sanofi-Aventis (FR) 2008-07-02 EP claimed
EP-2121635-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES Sanofi-Aventis (FR) 2009-11-25 EP disclosed
WO-2008078196-A2 SUBSTITUTED HETEROARYL PYRIDOPYRIMIDONE DERIVATIVES SANOFI-AVENTIS (FR) 2008-07-03 WO disclosed
EP-1939187-A1 Substituted heteroaryl pyridopyrimidone derivatives Sanofi-Aventis (FR) 2008-07-02 EP disclosed