SCHEMBL4390635

SCHEMBL4390635

O=C(c1ccccc1)c1ccc(CN(CCCN(Cc2ccccc2)C(=O)O)C(=O)OCc2scnc2C(=O)c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.39
BCHE P06276 4/20 0.39
ALDH1A1 P00352 2/20 0.36
HTT P42858 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP3A4 P08684 1/20 0.36
CCR6 P51684 1/20 0.36
PAX8 Q06710 1/20 0.36
SRD5A2 P31213 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL893102 0.91 HDAC3 (0.44) ACHEBCHEALDH1A1HTTSMN1; SMN2
SCHEMBL893528 0.90 CYP3A4 (0.47) CYP3A4RAB9A
SCHEMBL4390638 0.80 CYP3A4 (0.51) CYP3A4RAB9A
SCHEMBL4252383 0.80 TSHR (0.43) ACHEALDH1A1HTTL3MBTL1GAA
SCHEMBL4251206 0.79 ALOX5 (0.43) BCHEL3MBTL1
SCHEMBL893530 0.78 CYP3A4 (0.52) SMN1; SMN2CYP3A4RAB9A
SCHEMBL4248044 0.73 CYP3A4 (0.57) CYP3A4RAB9A
SCHEMBL4251210 0.72 CYP3A4 (0.51) L3MBTL1CYP3A4RAB9A
SCHEMBL9943426 0.72 CYP3A4 (0.54) CYP3A4
SCHEMBL893181 0.72 L3MBTL1 (0.44) ALDH1A1L3MBTL1HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP claimed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO claimed
EP-2465855-A1 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed
EP-2465856-A2 Cytochrome P450 oxidase inhibitors and uses thereof Abbott Laboratories (US) 2012-06-20 EP disclosed
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed