SCHEMBL4251206

SCHEMBL4251206

O=C(O)N(CCCN(Cc1ccc(OCc2ccccc2)cc1)C(=O)OCc1scnc1OCc1ccccc1)Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
MMP13 P45452 4/20 0.41
BCHE P06276 1/20 0.40
MMP2 P08253 1/20 0.40
PARP10 Q53GL7 1/20 0.39
LTA4H P09960 1/20 0.39
EPHX2 P34913 1/20 0.39
EPOR P19235 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL893517 0.90 CYP3A4 (0.48) ALOX5PTGS1PTGS2L3MBTL1MMP13
SCHEMBL4252383 0.88 TSHR (0.43) ALOX5L3MBTL1
SCHEMBL4251210 0.83 CYP3A4 (0.51) ALOX5PTGS1PTGS2L3MBTL1MMP13
SCHEMBL893518 0.81 CYP3A4 (0.53) ALOX5PTGS1PTGS2L3MBTL1MMP13
SCHEMBL893181 0.81 L3MBTL1 (0.44) L3MBTL1
SCHEMBL4390635 0.79 ACHE (0.39) L3MBTL1BCHE
SCHEMBL893827 0.79 CYP3A4 (0.48) PARP10
SCHEMBL23120532 0.75 LTA4H (0.64) ALOX5PTGS1PTGS2L3MBTL1BCHE
SCHEMBL4248044 0.73 CYP3A4 (0.57)
SCHEMBL23120176 0.72 ALOX5 (0.56) ALOX5PTGS1PTGS2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP claimed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO claimed