Benzamide

Benzamide

SCHEMBL4390826

NC(=O)c1ccccc1.N[C@@H](CS)C(=O)O

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.59
POLB P06746 1/20 0.59
CYP3A4 P08684 1/20 0.59
PARP1 P09874 1/20 0.59
MAPT P10636 1/20 0.59
TSHR P16473 1/20 0.59
CYP2C19 P33261 1/20 0.59
RECQL P46063 1/20 0.59
BLM P54132 1/20 0.59
PMP22 Q01453 1/20 0.59
HSD17B10 Q99714 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
SLC7A11 Q9UPY5 1/20 0.59
ALPI P09923 1/20 0.48
PKM P14618 1/20 0.48
XIAP P98170 1/20 0.48
SLC7A5 Q01650 1/20 0.48
KIF11 P52732 4/20 0.48
PLA2G10 O15496 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzophenone SCHEMBL29200984 0.87 PTGS1 (0.61) PTGS1TDP1L3MBTL1SLC7A11ALPI
Benzoic Acid SCHEMBL28091952 0.87 PTGS1 (0.61) PTGS1TSHRSLC7A11ALPIPKM
Benzil SCHEMBL5579330 0.87 PTGS1 (0.61) PTGS1SLC7A11ALPIPKMXIAP
Benzil SCHEMBL5579332 0.87 PTGS1 (0.61) PTGS1SLC7A11ALPIPKMXIAP
Benzoic Acid SCHEMBL28976988 0.84 PTGS1 (0.57) PTGS1TSHRSLC7A11ALPIPKM
Benzamide SCHEMBL6443169 0.83 TSHR (0.61) PTGS1POLBCYP3A4PARP1MAPT
Niacinamide SCHEMBL5946479 0.82 F7 (0.65) PTGS1CYP2C19TDP1SLC7A11
Biphenyl SCHEMBL27974455 0.82 PTGS1 (0.67) PTGS1SLC7A11ALPIPKMXIAP
Cysteine SCHEMBL28009382 0.82 PTGS1 (0.89) PTGS1BLMPMP22SLC7A11ALPI
Benzamide SCHEMBL28175463 0.81 TSHR (0.59) PTGS1POLBCYP3A4PARP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1435964-B1 NOVEL PRODRUGS OF N-H BOND-CONTAINING COMPOUNDS AND METHODS OF MAKING THEREOF UNIV KANSAS (US) 2009-12-09 EP disclosed
EP-1435964-A4 NOVEL PRODRUGS OF N-H BOND-CONTAINING COMPOUNDS AND METHODS OF MAKING THEREOF UNIV KANSAS (US) 2005-01-19 EP disclosed
EP-1435964-A2 NOVEL PRODRUGS OF N-H BOND-CONTAINING COMPOUNDS AND METHODS OF MAKING THEREOF The University of Kansas (US) 2004-07-14 EP disclosed
US-20030119814-A1 Novel prodrugs of N-H bond-containing compounds and methods of making thereof THE UNIVERSITY OF KANSAS 2003-06-26 US disclosed
WO-2003032908-A2 NOVEL PRODRUGS OF N-H BOND-CONTAINING COMPOUNDS AND METHODS OF MAKING THEREOF UNIVERSITY OF KANSAS (US) 2003-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030119814-A1 Novel prodrugs of N-H bond-containing compounds and methods of making thereof CTH, CBS, GSTP1 PTGS1 108/4885POLB 4177/4885CYP3A4 136/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.