Gw-328267

Gw-328267

SCHEMBL4390982

CCn1nnc([C@H]2O[C@@H](n3cnc4c(N)nc(NC(CO)Cc5ccccc5)nc43)[C@H](O)[C@@H]2O)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 1.00
ADORA3 P0DMS8 19/20 1.00
ADORA1 P30542 12/20 1.00
ADORA2B P29275 10/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gw-328267 SCHEMBL1980933 1.00 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL1979140 1.00 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL1983128 1.00 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL29369354 1.00 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL13268529 1.00 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL1983126 1.00 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL13268494 1.00 ADORA2A (1.00) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL5089293 0.99 ADORA2A (0.99) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL7228505 0.96 ADORA2A (0.93) ADORA2AADORA3ADORA1ADORA2B
Gw-328267 SCHEMBL7224617 0.96 ADORA2A (0.93) ADORA2AADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240358634-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS DOMPÉ FARMACEUTICI S.P.A. (IT) 2024-10-31 US disclosed
US-11969501-B2 Auris formulations for treating otic diseases and conditions DOMPÉ FARMACEUTICI S.P.A. (IT) 2024-04-30 US disclosed
US-11918653-B2 Triglyceride otic formulations and uses thereof DOMPÉ FARMACEUTICI S.P.A. (IT) 2024-03-05 US disclosed
US-20220040096-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS OTONOMY INC (US) 2022-02-10 US disclosed
US-20220040095-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS DOMPÉ FARMACEUTICI S.P.A. (IT) 2022-02-10 US disclosed
US-11123285-B2 Auris formulations for treating OTIC diseases and conditions OTONOMY, INC. (US) 2021-09-21 US disclosed
US-11123286-B2 Auris formulations for treating otic diseases and conditions OTONOMY, INC. (US) 2021-09-21 US disclosed
US-20210138069-A1 TRIGLYCERIDE OTIC FORMULATIONS AND USES THEREOF DOMPÉ FARMACEUTICI S.P.A. (IT) 2021-05-13 US disclosed
US-20200397907-A1 TRIGLYCERIDE OTIC FORMULATIONS AND USES THEREOF OTONOMY, INC. 2020-12-24 US disclosed
US-10751281-B2 Auris formulations for treating otic diseases and conditions OTONOMY, INC. (US) 2020-08-25 US disclosed
US-10272034-B2 Auris formulations for treating otic diseases and conditions OTONOMY, INC. (US) 2019-04-30 US disclosed
US-20180125781-A1 MODULATION OF GEL TEMPERATURE OF POLOXAMER-CONTAINING FORMULATIONS OTONOMY, INC. 2018-05-10 US disclosed
WO-2018005830-A1 TRIGLYCERIDE OTIC FORMULATIONS AND USES THEREOF OTONOMY, INC. (US) 2018-01-04 WO disclosed
US-20160243028-A1 Auris Formulations for Treating Otic Diseases and Conditions DOMPÉ FARMACEUTICI S.P.A. (IT) 2016-08-25 US disclosed
US-20160228357-A1 Auris Formulations for Treating Otic Diseases and Conditions OTONOMY, INC. 2016-08-11 US disclosed
US-20160095902-A1 Auris Formulations for Treating Otic Diseases and Conditions OTONOMY, INC. 2016-04-07 US disclosed
US-9132087-B2 Auris formulations for treating otic diseases and conditions OTONOMY, INC. (US) 2015-09-15 US disclosed
US-20120277199-A1 Modulation of Gel Temperature of Poloxamer-Containing Formulations OTONOMY, INC. (US) 2012-11-01 US disclosed
EP-2490722-A2 MODULATION OF GEL TEMPERATURE OF POLOXAMER-CONTAINING FORMULATIONS Otonomy, Inc. (US) 2012-08-29 EP disclosed
US-20090306225-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS OTONOMY, INC. (US) 2009-12-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (17 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180125781-A1 MODULATION OF GEL TEMPERATURE OF POLOXAMER-CONTAINING FORMULATIONS PTGIR, HSPH1, HSP90AA1 ADORA2A 1279/4885ADORA3 3154/4885ADORA1 2686/4885
US-20210138069-A1 TRIGLYCERIDE OTIC FORMULATIONS AND USES THEREOF CETP, LIPA, APOB ADORA2A 2398/4885ADORA3 2478/4885ADORA1 2255/4885
US-20160243028-A1 Auris Formulations for Treating Otic Diseases and Conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-20220040096-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-11123286-B2 Auris formulations for treating otic diseases and conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-10751281-B2 Auris formulations for treating otic diseases and conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-20090306225-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-20160095902-A1 Auris Formulations for Treating Otic Diseases and Conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-11123285-B2 Auris formulations for treating OTIC diseases and conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-11918653-B2 Triglyceride otic formulations and uses thereof CETP, LIPA, APOB ADORA2A 2398/4885ADORA3 2478/4885ADORA1 2255/4885
US-10272034-B2 Auris formulations for treating otic diseases and conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-20160228357-A1 Auris Formulations for Treating Otic Diseases and Conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-20240358634-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-20120277199-A1 Modulation of Gel Temperature of Poloxamer-Containing Formulations PTGIR, HSPH1, HSP90AA1 ADORA2A 1279/4885ADORA3 3154/4885ADORA1 2686/4885
US-20200397907-A1 TRIGLYCERIDE OTIC FORMULATIONS AND USES THEREOF CETP, LIPA, APOB ADORA2A 2246/4885ADORA3 2382/4885ADORA1 2143/4885
US-20220040095-A1 AURIS FORMULATIONS FOR TREATING OTIC DISEASES AND CONDITIONS OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885
US-11969501-B2 Auris formulations for treating otic diseases and conditions OTC, AQP4, SLC26A4 ADORA2A 24/4885ADORA3 84/4885ADORA1 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.