SCHEMBL4392216

SCHEMBL4392216

CCOc1ccc2c(c1)c(C(=O)C(=O)Nc1ccc(Cl)cc1)c(Cl)n2Cc1ccc(Cl)cc1Cl.COc1ccc2c(c1)c(C(=O)C(=O)Nc1ccc(Cl)cc1)c(Cl)n2Cc1ccc(Cl)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
POLB P06746 1/20 0.44
FAAH O00519 1/20 0.44
PLA2G2A P14555 2/20 0.42
PTGS2 P35354 3/20 0.42
KCNH2 Q12809 1/20 0.41
EDNRB P24530 3/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RGS12 O14924 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4089939 0.97 MEN1 (0.45) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL4088405 0.97 MEN1 (0.47) KMT2AMEN1NPC1RAB9APOLB
SCHEMBL4098796 0.95 KMT2A (0.46) KMT2AMEN1NPC1RAB9AFAAH
SCHEMBL4089993 0.93 KMT2A (0.48) KMT2AMEN1NPC1RAB9AFAAH
SCHEMBL3006768 0.93 PTGS2 (0.49) FAAHPLA2G2APTGS2EDNRBMAPT
SCHEMBL3010596 0.91 MEN1 (0.43) KMT2AMEN1POLBFAAHEDNRB
SCHEMBL4088721 0.90 KCNH2 (0.48) KMT2AMEN1NPC1RAB9AFAAH
SCHEMBL2999278 0.90 FAAH (0.44) KMT2AMEN1POLBFAAHTAS1R3
SCHEMBL3001524 0.90 PLA2G2A (0.46) KMT2AMEN1NPC1RAB9AFAAH
SCHEMBL4378535 0.90 FAAH (0.52) KMT2AMEN1NPC1RAB9AFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049520-A2 INDOLE COMPOUNDS Ironwood Pharmaceuticals, Inc. (US) 2009-04-22 EP disclosed
WO-2008019357-A2 INDOLE COMPOUNDS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed