SCHEMBL4392568

SCHEMBL4392568

Clc1cc2c(N3CCOCC3)nc(CN3CCNCC3)cc2s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
CSF1R P07333 1/20 0.35
PIM1 P11309 1/20 0.35
PIM2 Q9P1W9 1/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PIK3CA P42336 4/20 0.35
PIK3CB P42338 1/20 0.35
CXCR4 P61073 2/20 0.35
PIK3R1 P27986 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
SOS1 Q07889 1/20 0.34
MAPT P10636 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
KDM5C P41229 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
JAK2 O60674 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10276093 0.92 RAB9A (0.41) RAB9ANPC1CSF1RPIM1PIM2
SCHEMBL3787431 0.88 CYP2D6 (0.37) KMT2AMEN1RAB9ANPC1CSF1R
SCHEMBL10275931 0.84 HRH3 (0.44) PIK3CAPIK3CB
SCHEMBL3782027 0.84 LGMN (0.35) KMT2AMEN1RAB9ANPC1CSF1R
SCHEMBL10276136 0.83 HRH3 (0.38) RAB9ANPC1TSHRPIK3CAPIK3CB
SCHEMBL10276385 0.82 PIK3CD (0.47) PIK3CAPIK3CB
SCHEMBL3778364 0.81 SMN1; SMN2 (0.38) RAB9ANPC1TSHRPIK3CAPIK3R1
SCHEMBL4554726 0.81 SMN1; SMN2 (0.38) RAB9ANPC1TSHRPIK3CAPIK3R1
SCHEMBL14955228 0.80 PIK3CA (0.41) PIK3CAPIK3CBPIK3R1SMN1; SMN2
SCHEMBL3809370 0.80 HRH3 (0.37) PIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041139-A2 PHARMACEUTICAL COMPOUNDS F.HOFFMANN-LA ROCHE AG (CH) 2009-04-01 EP disclosed
WO-2007127175-A2 PHARMACEUTICAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2007-11-08 WO disclosed