SCHEMBL4392758

SCHEMBL4392758

FC1=C(CCI)C(F)(F)C1(F)F

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250963 0.69
SCHEMBL333168 0.61
SCHEMBL3834726 0.58
SCHEMBL30899713 0.55
SCHEMBL7331916 0.53 SLC6A2 (0.31)
SCHEMBL10685237 0.53 ALDH1A1 (0.30)
SCHEMBL251017 0.49
SCHEMBL2137807 0.49
SCHEMBL2137624 0.49
SCHEMBL252349 0.49

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090306297-A1 PROCESS FOR PREPARING A COPOLYMER WITH CONTROLLED ARCHITECTURE, OF TELOMER OR BLOCK COPOLYMER TYPE, OBTAINED FROM VINYL PHOSPHONATE MONOMERS, BY IODINE TRANSFER POLYMERIZATION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2009-12-10 US claimed
EP-1976888-B1 PROCESS FOR PREPARING A COPOLYMER WITH CONTROLLED ARCHITECTURE, OF TELOMER OR BLOCK COPOLYMER TYPE, OBTAINED FROM VINYL PHOSPHONATE MONOMERS, BY IODINE TRANSFER POLYMERIZATION RHODIA OPERATIONS (FR) 2012-06-13 EP disclosed
US-20090306297-A1 PROCESS FOR PREPARING A COPOLYMER WITH CONTROLLED ARCHITECTURE, OF TELOMER OR BLOCK COPOLYMER TYPE, OBTAINED FROM VINYL PHOSPHONATE MONOMERS, BY IODINE TRANSFER POLYMERIZATION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2009-12-10 US disclosed
EP-1976888-A1 PROCESS FOR PREPARING A COPOLYMER WITH CONTROLLED ARCHITECTURE, OF TELOMER OR BLOCK COPOLYMER TYPE, OBTAINED FROM VINYL PHOSPHONATE MONOMERS, BY IODINE TRANSFER POLYMERIZATION Rhodia Opérations (FR) 2008-10-08 EP disclosed
WO-2007085623-A1 PROCESS FOR PREPARING A COPOLYMER WITH CONTROLLED ARCHITECTURE, OF TELOMER OR BLOCK COPOLYMER TYPE, OBTAINED FROM VINYL PHOSPHONATE MONOMERS, BY IODINE TRANSFER POLYMERIZATION RHODIA OPERATIONS (FR) 2007-08-02 WO disclosed
EP-0759447-B1 Fluorine containing rubbers, process for their preparation, process for the preparation of fluoroelastomers and their use BAYER AG (DE) 2002-07-17 EP disclosed
EP-0759447-A2 Fluorine containing rubbers, process for their preparation, process for the preparation of fluoroelastomers and their use BAYER AG (DE) 1997-02-26 EP disclosed
EP-0489370-B1 Process for preparing polymer DAIKIN IND LTD (JP) 1997-02-05 EP disclosed
US-5439980-A In presence of a free radical catalyst and an iodide DAIKIN INDUSTRIES (JP) 1995-08-08 US disclosed
EP-0489370-A1 Process for preparing polymer DAIKIN INDUSTRIES, LIMITED (JP) 1992-06-10 EP disclosed