SCHEMBL4396358

SCHEMBL4396358

CCn1cc(C(=O)O)c(=O)c2cc(SCCNCCNC(=O)OC(C)(C)C)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.48
KDM4E B2RXH2 7/20 0.48
HPGD P15428 7/20 0.48
HSD17B10 Q99714 5/20 0.48
TSHR P16473 3/20 0.48
RAB9A P51151 1/20 0.48
LMNA P02545 7/20 0.43
HTT P42858 4/20 0.43
TDP1 Q9NUW8 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
APEX1 P27695 1/20 0.42
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
MAPK1 P28482 1/20 0.39
DRD3 P35462 1/20 0.38
POLB P06746 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3983498 0.94 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL3983514 0.94 ALDH1A1 (0.51) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL3811662 0.91 LMNA (0.52) ALDH1A1KDM4EHPGDHSD17B10TSHR
Formic Acid SCHEMBL4392627 0.88 LMNA (0.49) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL3812384 0.87 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL3983501 0.86 LMNA (0.42) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL3816675 0.85 LMNA (0.55) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL4541684 0.85 KDM4E (0.57) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL5471995 0.83 LMNA (0.42) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL4392504 0.82 ALDH1A1 (0.48) ALDH1A1KDM4EHPGDHSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628990-B1 NOVEL 14 AND 15 MEMBERED RING COMPOUNDS GLAXO GROUP LTD (GB) 2009-12-02 EP disclosed
US-20070141276-A1 Novel 14 and 15 membered ring compounds GLAXO GROUP LIMITED (GB) 2007-06-21 US disclosed
CN-1816557-A Novel 14 and 15 membered ring compounds GLAXO GROUP LTD (GB) 2006-08-09 CN disclosed