SCHEMBL4396938

SCHEMBL4396938

O=C(NO)c1cccc(B(O)O)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.61
HDAC1 Q13547 5/20 0.61
KDM4E B2RXH2 1/20 0.58
EGLN2 Q96KS0 1/20 0.58
HDAC8 Q9BY41 9/20 0.56
HDAC2 Q92769 5/20 0.52
HDAC3 O15379 3/20 0.52
HDAC7 Q8WUI4 2/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
IDO1 P14902 1/20 0.52
ALOX15 P16050 1/20 0.52
CA9 Q16790 1/20 0.52
HSD17B10 Q99714 1/20 0.52
NCOR2 Q9Y618 1/20 0.52
ENPP2 Q13822 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL190230 0.83 HDAC6 (0.59) HDAC6HDAC1KDM4EHDAC8HDAC2
SCHEMBL29956030 0.83 ALDH1A1 (0.59) HDAC6HDAC1KDM4ECA1ENPP2
SCHEMBL1445203 0.83 ALDH1A1 (0.59) HDAC6HDAC1KDM4ECA1ENPP2
Hydrochloric Acid SCHEMBL4551090 0.81 ALDH1A1 (0.58) HDAC6HDAC1KDM4ECA1ENPP2
SCHEMBL11791484 0.81 HDAC8 (0.79) HDAC6HDAC1KDM4EEGLN2HDAC8
SCHEMBL3756621 0.79 ENPP2 (0.47) KDM4EENPP2
SCHEMBL1933481 0.79 HDAC1 (0.63) HDAC6HDAC1HDAC8HDAC2
SCHEMBL520859 0.79 LMNA (0.49)
SCHEMBL177725 0.79 NPSR1 (0.56) KDM4EHSD17B10ENPP2
SCHEMBL3031782 0.79 SMN1; SMN2 (0.50) HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed