SCHEMBL4397164

SCHEMBL4397164

CCOC(=O)c1ccc(C(=O)NO)cc1F

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.58
HDAC6 Q9UBN7 4/20 0.58
TDP1 Q9NUW8 2/20 0.48
POLB P06746 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KDM4E B2RXH2 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CA12 O43570 3/20 0.45
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45
CA7 P43166 3/20 0.45
CA9 Q16790 3/20 0.45
CA14 Q9ULX7 3/20 0.45
TSHR P16473 1/20 0.45
NPC1 O15118 1/20 0.44
MEN1 O00255 2/20 0.43
MAPT P10636 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7222675 0.81 TSHR (0.53) TDP1POLBSMN1; SMN2KDM4ELMNA
SCHEMBL11706325 0.79 CA12 (0.45) KDM4ELMNACA12CA1CA2
SCHEMBL6676941 0.79 TRPA1 (0.47) HDAC6TDP1POLBSMN1; SMN2KDM4E
SCHEMBL719657 0.78 DGAT1 (0.54) SMN1; SMN2LMNACA12CA1CA2
SCHEMBL19203928 0.78 CA12 (0.50) LMNAHTTCA12CA1CA2
SCHEMBL367075 0.78 TSHR (0.57) TDP1POLBSMN1; SMN2NPSR1CA12
Hydrochloric Acid SCHEMBL31426389 0.77 DGAT1 (0.53) SMN1; SMN2LMNACA12CA1CA2
SCHEMBL1353042 0.77 CA12 (0.54) POLBSMN1; SMN2KDM4ELMNATP53
SCHEMBL6675739 0.77 SMN1; SMN2 (0.44) TDP1POLBSMN1; SMN2KDM4ELMNA
SCHEMBL927276 0.76 CA12 (0.70) LMNATP53CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed