SCHEMBL4397407

SCHEMBL4397407

N=C(NN)c1ccc2c(c1)NC(=O)C2

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 8/20 0.52
CRBN Q96SW2 2/20 0.51
AHR P35869 3/20 0.49
CMA1 P23946 2/20 0.49
EIF2AK2 P19525 1/20 0.47
PDK2 Q15119 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.40
TDP2 O95551 1/20 0.40
EPHX2 P34913 1/20 0.39
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzamidine SCHEMBL4399664 0.90 SMYD3 (0.45) SMYD3CRBNAHRCMA1EIF2AK2
SCHEMBL4394998 0.88 SMYD3 (0.52) SMYD3AHRHDAC3EPHX2
Hydrochloric Acid SCHEMBL4399720 0.87 SMYD3 (0.51) SMYD3AHRHDAC3EPHX2
SCHEMBL4398573 0.86 AHR (0.54) SMYD3CRBNAHRCMA1EIF2AK2
SCHEMBL30760741 0.79 SMYD3 (0.58) SMYD3CRBNAHRCMA1EIF2AK2
SCHEMBL3194345 0.79 SMYD3 (0.58) SMYD3CRBNAHRCMA1EIF2AK2
Hydrochloric Acid SCHEMBL29528151 0.78 SMYD3 (0.57) SMYD3CRBNAHRCMA1EIF2AK2
SCHEMBL29713338 0.76 TDP2 (0.66) SMYD3CRBNAHRCMA1EIF2AK2
SCHEMBL398818 0.76 TDP2 (0.66) SMYD3CRBNAHRCMA1EIF2AK2
SCHEMBL24124675 0.74 AHR (0.59) SMYD3CRBNAHRCMA1EIF2AK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101321525-B Heteroaryl substituted piperidine derivatives as L-CPT1 inhibitors HOFFMANN LA ROCHE 2013-01-30 CN disclosed
EP-1959951-B1 HETEROARYL SUBSTITUTED PIPERIDINE DERIVATIVES AS L-CPT1 INHIBITORS HOFFMANN LA ROCHE (CH) 2009-12-23 EP disclosed