SCHEMBL4398637

SCHEMBL4398637

O=C(O)c1ccccc1-c1ccc(/C=C2\SC(=S)N(Cc3ccccc3)C2=O)o1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 1.00
SYK P43405 1/20 0.81
MEN1 O00255 6/20 0.72
KMT2A Q03164 6/20 0.72
POLB P06746 5/20 0.72
ALDH1A1 P00352 4/20 0.72
MAPT P10636 4/20 0.72
MCL1 Q07820 3/20 0.72
RECQL P46063 3/20 0.72
NPSR1 Q6W5P4 2/20 0.72
TDP1 Q9NUW8 2/20 0.72
EIF4E P06730 1/20 0.72
EIF4G1 Q04637 1/20 0.72
THRB P10828 1/20 0.72
MAP3K5 Q99683 7/20 0.65
LMNA P02545 2/20 0.64
ALOX12 P18054 2/20 0.64
NPC1 O15118 1/20 0.61
RAB9A P51151 1/20 0.61
PTP4A3 O75365 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4402019 1.00 ENPP2 (1.00) ENPP2SYKMEN1KMT2APOLB
SCHEMBL1135868 0.90 SYK (1.00) ENPP2SYKMEN1KMT2APOLB
SCHEMBL12668370 0.90 SYK (1.00) ENPP2SYKMEN1KMT2APOLB
SCHEMBL30774050 0.90 SYK (1.00) ENPP2SYKMEN1KMT2APOLB
SCHEMBL1135867 0.90 SYK (1.00) ENPP2SYKMEN1KMT2APOLB
SCHEMBL3796210 0.89 ENPP2 (0.80) ENPP2SYKMEN1KMT2APOLB
SCHEMBL29987110 0.89 ENPP2 (0.80) ENPP2SYKMEN1KMT2APOLB
SCHEMBL3796207 0.89 ENPP2 (0.80) ENPP2SYKMEN1KMT2APOLB
SCHEMBL8337281 0.88 ENPP2 (0.78) ENPP2SYKMEN1KMT2APOLB
SCHEMBL3897831 0.87 MAP3K5 (0.78) ENPP2SYKMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1830848-B1 USE OF THIAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF SOLID TUMORS CELL THERAPEUTICS EUROPE SRL (IT) 2009-12-16 EP claimed
US-20080261980-A1 Use of Thiazolidinone Derivatives as Antiangiogenic Agents CELL THERAPEUTICS, INC. (US) 2008-10-23 US claimed
WO-2020236668-A1 LEUKADHERIN-1 ALONE OR IN COMBINATION FOR USE IN THE TREATMENT OF CANCER GB006, INC. (US) 2020-11-26 WO disclosed
EP-1830848-B1 USE OF THIAZOLIDINONE DERIVATIVES FOR THE TREATMENT OF SOLID TUMORS CELL THERAPEUTICS EUROPE SRL (IT) 2009-12-16 EP disclosed
US-20080261980-A1 Use of Thiazolidinone Derivatives as Antiangiogenic Agents CELL THERAPEUTICS, INC. (US) 2008-10-23 US disclosed
EP-1830848-A1 USE OF THIAZOLIDINONE DERIVATIVES AS ANTIANGIOGENIC AGENTS Cell Therapeutics Europe S.R.L. (IT) 2007-09-12 EP disclosed
WO-2006066846-A1 USE OF THIAZOLIDINONE DERIVATIVES AS ANTIANGIOGENIC AGENTS CELL THERAPEUTICS EUROPE S.R.L. (IT) 2006-06-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080261980-A1 Use of Thiazolidinone Derivatives as Antiangiogenic Agents EP300, HIF1A, HIF1AN ENPP2 2878/4885SYK 3137/4885MEN1 2216/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.