SCHEMBL4400715

SCHEMBL4400715

Cc1cc[n+](CCCc2ccc(-c3ccc(CCC[n+]4ccc(C)cc4)cc3)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.68
CHRNA10 Q9GZZ6 2/20 0.68
CHRNA9 Q9UGM1 2/20 0.68
CHKA P35790 3/20 0.57
HTT P42858 3/20 0.53
KDM4E B2RXH2 2/20 0.46
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MEN1 O00255 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP1A2 P05177 2/20 0.45
TP53 P04637 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAPK1 P28482 1/20 0.44
RAD52 P43351 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4405443 0.89 HTT (0.61) CHRNA7CHRNA10CHRNA9CHKAHTT
SCHEMBL13334229 0.88 CHRNA7 (0.55) CHRNA7CHRNA10CHRNA9CHKAHTT
Bromide SCHEMBL3313967 0.87 CHRNA7 (0.56) CHRNA7CHRNA10CHRNA9CHKAHTT
SCHEMBL5292316 0.86 KDM4E (0.53) CHRNA7CHRNA10CHRNA9CHKAHTT
SCHEMBL13334099 0.82 HTT (0.69) CHRNA7CHRNA10CHRNA9CHKAHTT
SCHEMBL4404376 0.82 CHKA (0.65) CHRNA7CHRNA10CHRNA9CHKAHTT
Bromide SCHEMBL3314015 0.81 HTT (0.67) CHRNA7CHRNA10CHRNA9CHKAHTT
SCHEMBL4398944 0.81 CHRNA7 (1.00) CHRNA7CHRNA10CHRNA9CHKAHTT
SCHEMBL13361695 0.80 HTT (0.60) CHRNA7CHRNA10CHRNA9CHKAHTT
SCHEMBL4403538 0.80 HTT (0.50) CHRNA7CHRNA10CHRNA9CHKAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178678-B2 Bis-quaternary ammonium salts and methods for modulating neuronal nicotinic acetylcholine receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2012-05-15 US disclosed
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2010-03-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors CHRNA2, CHRNA5, CHRNA4 CHRNA7 7/4885CHRNA10 4/4885CHRNA9 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.