SCHEMBL4404376

SCHEMBL4404376

Cc1cc[n+](CCc2ccc(CC[n+]3ccc(C)cc3)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHKA P35790 6/20 0.65
HTT P42858 2/20 0.50
CYP1A2 P05177 1/20 0.46
CYP2A6 P11509 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
CHRNA7 P36544 2/20 0.46
CHRNA10 Q9GZZ6 2/20 0.46
CHRNA9 Q9UGM1 2/20 0.46
KCNH2 Q12809 1/20 0.42
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
RAD52 P43351 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
IDO1 P14902 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13838215 0.89 CHKA (0.53) CHKAHTTTAAR1KCNH2KDM4E
SCHEMBL13361695 0.88 HTT (0.60) CHKAHTTCYP1A2CHRNA7CHRNA10
Hydrochloric Acid SCHEMBL10935706 0.87 ALDH1A1 (0.55) CHKAHTTKCNH2KDM4EALDH1A1
Bromide SCHEMBL8857808 0.87 CHKA (0.57) CHKAHTTMEN1KMT2AKDM4E
SCHEMBL4405443 0.84 HTT (0.61) CHKAHTTCHRNA7CHRNA10CHRNA9
Hydrochloric Acid SCHEMBL11281826 0.83 CHKA (0.48) CHKAHTTMEN1MAPTKMT2A
SCHEMBL4400715 0.82 CHRNA7 (0.68) CHKAHTTCYP1A2CYP2A6TAAR1
SCHEMBL2610346 0.82 CHKA (0.47) CHKAHTTCYP1A2CYP2A6TAAR1
SCHEMBL21290572 0.81 HTT (0.61) CHKAHTTCYP1A2MEN1MAPT
SCHEMBL10188714 0.78 CHRNA7 (0.73) CHKACHRNA7CHRNA10CHRNA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178678-B2 Bis-quaternary ammonium salts and methods for modulating neuronal nicotinic acetylcholine receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2012-05-15 US disclosed
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 2010-03-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100069432-A1 Bis-Quaternary Ammonium Salts and Methods for Modulating Neuronal Nicotinic Acetylcholine Receptors CHRNA2, CHRNA5, CHRNA4 CHKA 332/4885HTT 603/4885CYP1A2 2739/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.