SCHEMBL4403749

SCHEMBL4403749

CC(=O)c1ccc2ccc(N)nc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 3/20 0.52
BACE1 P56817 3/20 0.48
CYP2A6 P11509 1/20 0.46
CA2 P00918 1/20 0.44
NCF1 P14598 6/20 0.44
NOS2 P35228 1/20 0.44
MAPT P10636 2/20 0.43
PRKCI P41743 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
NCK1 P16333 1/20 0.43
CREBBP Q92793 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
TNNI3 P19429 1/20 0.40
TNNT2 P45379 1/20 0.40
RAB9A P51151 1/20 0.40
TNNC1 P63316 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4403751 0.87 BACE1 (0.55) PLAUBACE1CYP2A6CA2NCF1
SCHEMBL2671555 0.83 PLAU (0.57) PLAUBACE1NCF1NOS2MAPT
SCHEMBL15043775 0.81 CYP2A6 (0.46) CYP2A6CA2MAPTALDH1A1HPGD
SCHEMBL4145913 0.81 PLAU (0.49) PLAUBACE1NCF1NOS2NCK1
SCHEMBL16947985 0.81 PLAU (0.52) PLAUBACE1CA2NCF1MAPT
SCHEMBL9015187 0.79 CYP1A2 (0.53) CYP2A6MAPTALDH1A1HPGDMEN1
SCHEMBL10151651 0.77 MAP4K4 (0.42) CYP2A6CA2MAPTPRKCIALDH1A1
SCHEMBL4407433 0.76 NCF1 (0.48) CYP2A6NCF1MAPTPRKCIALDH1A1
SCHEMBL4410086 0.75 MTNR1A (0.54) CYP2A6MAPTALDH1A1HPGDKDM4E
SCHEMBL9015204 0.74 CYP2A6 (0.42) CYP2A6MAPTALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed