SCHEMBL4410086

SCHEMBL4410086

COc1ccc2ccc(C(C)=O)cc2n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.54
MTNR1B P49286 1/20 0.54
CYP2A6 P11509 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HPGD P15428 2/20 0.41
NNMT P40261 2/20 0.41
MAPT P10636 2/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2671576 0.86 KDM4E (0.54) MTNR1AMTNR1BALDH1A1KMT2AGAA
SCHEMBL4137126 0.82 MTNR1A (0.47) MTNR1AMTNR1BALDH1A1HDAC3HDAC4
SCHEMBL2671191 0.80 HSD17B2 (0.52) MTNR1AMTNR1BALDH1A1KMT2AMAPT
SCHEMBL25804157 0.79 HPGD (0.46) ALDH1A1KMT2AHPGDNNMTMAPT
SCHEMBL30134289 0.79 HPGD (0.46) ALDH1A1KMT2AHPGDNNMTMAPT
SCHEMBL30133957 0.79 SMN1; SMN2 (0.44) ALDH1A1KMT2AHPGDNNMTMAPT
SCHEMBL9015187 0.77 CYP1A2 (0.53) CYP2A6ALDH1A1KMT2AHPGDMAPT
SCHEMBL8148257 0.76 CYP2A6 (0.44) CYP2A6ALDH1A1KMT2AGAAHPGD
SCHEMBL8156878 0.76 ALDH1A1 (0.43) CYP2A6ALDH1A1KMT2AGAAHPGD
SCHEMBL4403749 0.75 PLAU (0.52) CYP2A6ALDH1A1KMT2AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012056372-A1 N1/N2-LACTAM ACETYL-CoA CARBOXYLASE INHIBITORS PFIZER INC. (US) 2012-05-03 WO disclosed