SCHEMBL4405573

SCHEMBL4405573

CC(C)COc1cccc2[nH]c(OC(=O)Nc3ccc(CN(C)C4CCOCC4)cc3)cc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.42
CCR2 P41597 3/20 0.39
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
LMNA P02545 2/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 3/20 0.35
NPC1 O15118 1/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
ADRB3 P13945 4/20 0.34
PTGER1 P34995 1/20 0.34
CYP2D6 P10635 2/20 0.34
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
HDAC1 Q13547 1/20 0.34
MLNR O43193 1/20 0.34
NR1I2 O75469 1/20 0.34
ADRB2 P07550 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4400749 0.88 PTGER1 (0.34) MEN1KMT2ALMNAALDH1A1MAPT
SCHEMBL914650 0.87 MEN1 (0.47) CCR5CCR2MEN1KMT2ALMNA
SCHEMBL4411253 0.81 LMNA (0.35) LMNAALDH1A1MAPTNPC1RAB9A
SCHEMBL4409139 0.76 ADRB3 (0.41) MEN1KMT2AADRB3PTGER1
SCHEMBL914632 0.75 KMT2A (0.47) MEN1KMT2ALMNAALDH1A1MAPT
SCHEMBL914267 0.71 KDM4E (0.38) MEN1KMT2ALMNAALDH1A1NPC1
SCHEMBL6963102 0.71 KDM4E (0.38) MEN1KMT2ALMNAALDH1A1NPC1
SCHEMBL12905932 0.70 KMT2A (0.38) MEN1KMT2ALMNAALDH1A1NPC1
SCHEMBL17571837 0.68 NPC1 (0.53) CCR5CCR2LMNAALDH1A1NPC1
SCHEMBL7216495 0.68 CCR5 (0.52) CCR5CCR2ALDH1A1MAPTCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720859-B1 CHEMOKINE RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2009-12-23 EP claimed