SCHEMBL4407004

SCHEMBL4407004

NCc1cccc(C2(O)CCN(C(=O)O)CC2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
OPRL1 P41146 2/20 0.47
POLB P06746 1/20 0.46
ALDH1A1 P00352 3/20 0.45
PARP10 Q53GL7 1/20 0.45
NOS2 P35228 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CHRM4 P08173 2/20 0.43
SIGMAR1 Q99720 1/20 0.43
LMNA P02545 1/20 0.41
OPRM1 P35372 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368267 0.87 ALDH1A1 (0.47) MEN1KMT2AOPRL1POLBALDH1A1
SCHEMBL4412901 0.81 OPRD1 (0.51) ALDH1A1NOS2CHRM4CYP4F2CYP4A11
SCHEMBL301794 0.80 OPRL1 (0.75) KMT2AOPRL1POLBALDH1A1SIGMAR1
SCHEMBL795975 0.80 ALDH1A1 (0.56) MEN1KMT2AOPRL1POLBALDH1A1
SCHEMBL3441859 0.79 OPRM1 (0.60) MEN1KMT2AOPRL1ALDH1A1LMNA
SCHEMBL5373048 0.79 OPRM1 (0.60) MEN1KMT2AOPRL1POLBALDH1A1
SCHEMBL19280276 0.79 ALDH1A1 (0.46) OPRL1ALDH1A1PARP10CA12CA1
SCHEMBL2931056 0.79 OPRM1 (0.52) MEN1KMT2AOPRL1ALDH1A1LMNA
SCHEMBL2587746 0.79 ALDH1A1 (0.50) OPRL1ALDH1A1NOS2OPRM1CYP4F2
SCHEMBL14696653 0.79 PTPN1 (0.48) MEN1KMT2AOPRL1POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-B1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMA INC (US) 2009-12-23 EP disclosed