SCHEMBL4407407

SCHEMBL4407407

COC(=O)C1=C(C)Nc2cc[nH]c(=O)c2C1c1ccccc1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.56
NR1I2 O75469 1/20 0.51
POLB P06746 1/20 0.46
LMNA P02545 2/20 0.45
ACHE P22303 2/20 0.44
HSD17B10 Q99714 6/20 0.44
KDM4E B2RXH2 4/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2C9 P11712 3/20 0.44
CYP2C19 P33261 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TP53 P04637 2/20 0.44
MAPT P10636 2/20 0.44
CYP1A2 P05177 2/20 0.44
TSHR P16473 2/20 0.44
PDE1C Q14123 1/20 0.44
ABCC4 O15439 1/20 0.44
PLIN1 O60240 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10784001 0.90 ACHE (0.55) PKMPOLBLMNAACHEHSD17B10
SCHEMBL10784036 0.87 CYP2C9 (0.44) PKMNR1I2POLBLMNAHSD17B10
SCHEMBL10785934 0.87 NR1I2 (0.46) PKMNR1I2LMNAACHEHSD17B10
SCHEMBL10785872 0.84 CYP1A2 (0.58) NR1I2ACHEKDM4ECYP3A4CYP2C9
SCHEMBL10790585 0.84 ADORA3 (0.55) POLBACHEHSD17B10KDM4EALDH1A1
SCHEMBL10789033 0.83 ADORA3 (0.69) NR1I2POLBLMNAACHEHSD17B10
SCHEMBL31295852 0.83 NR3C2 (0.47) PKMNR1I2POLBHSD17B10KDM4E
SCHEMBL10786737 0.83 ALDH1A1 (0.60) PKMNR1I2POLBLMNAHSD17B10
SCHEMBL10789570 0.82 HSD17B10 (0.46) PKMNR1I2POLBLMNAHSD17B10
SCHEMBL10784567 0.81 ALDH1A1 (0.47) PKMNR1I2POLBLMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056934-A1 1,4-DIHYDRONAPHTHYRIDINE DERIVATIVES PFIZER PRODUCTS INC. (US) 2009-05-07 WO disclosed